VDM 11 (in Tocrisolve™ 100)

Discontinued Product

VDM 11 (in Tocrisolve™ 100) (Cat. No. 1686) has been withdrawn from sale for commercial reasons.
Cat.No. 1686 - VDM 11 (in Tocrisolve 100) | C27H39NO2 | CAS No. 313998-81-1
Description: Potent, selective anandamide transport inhibitor (in water-soluble emulsion)
Chemical Name: (5Z,8Z,11Z,14Z)-N-(4-Hydroxy-2-methylphenyl)-5,8,11,14-eicosatetraenamide
Datasheet
Citations
Reviews
Literature (3)

Biological Activity

A potent and selective inhibitor of the anandamide membrane transporter (AMT), in water-soluble emulsion (for details see TocrisoveTM 100). IC50 values for inhibition of AMT are 4 - 11 mM. Displays negligible agonist activity at the hVR1 receptor and very weak action at CB1 and CB2 receptors. Ki values are > 5 - 10 mM at CB1 and CB2. Active in vivo.

VDM 11, pure oil dissolved in ethanol and Tocrisolve Control also available.

Technical Data

M. Wt 409.61
Formula C27H39NO2
Storage Store at +4°C
CAS Number 313998-81-1
PubChem ID 9887748
InChI Key WUZWFRWVRHLXHZ-ZKWNWVNESA-N
Smiles O=C(NC1=C(C)C=C(O)C=C1)CCC\C=C/C\C=C/C/C=C\C/C=C\CCCCC

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for VDM 11 (in Tocrisolve™ 100)

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