Submit a Review & Earn an Amazon Gift Card
You can now submit reviews for your favorite Tocris products. Your review will help other researchers decide on the best products for their research. Why not submit a review today?!
Submit ReviewBiological Activity for Tertiapin LQ
Tertiapin LQ is a blocker of Kir1.1 channels; displays >250-fold selectivity for Kir1.1 (Kd values are 1.1, 274 and 361 nM for Kir1.1, Kir3.1/3.2 and Kir3.1/3.4 respectively). Derivative of tertiapin-Q (Cat. No. 1316).
Technical Data for Tertiapin LQ
| M. Wt | 2428.03 |
| Formula | C106H179N33O24S4 |
| Sequence |
ALCNCNRIIIPLQCWKKCGKK (Modifications: Disulfide bridge between 3 - 14, 5 - 18, Lys-21 = C-terminal amide) |
| Storage | Store at -20°C |
| PubChem ID | 90488935 |
| InChI Key | WUMIWMIQOSXVPZ-ZPWFPUPGSA-N |
| Smiles | [H]N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H]1CSSC[C@@H]2NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]3CCCN3C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC3=CNC4=C3C=CC=C4)NC2=O)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@H](CC(N)=O)NC1=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Solubility Data for Tertiapin LQ
| Solubility | Soluble to 2 mg/ml in 20% acetonitrile / water |
Product Datasheets for Tertiapin LQ
References for Tertiapin LQ
References are publications that support the biological activity of the product.
Ramu et al (2008) Engineered specific and high-affinity inhibitor for a subtype of inward-rectifier K+ channels. Proc.Natl.Acad.Sci.USA 105 10774 PMID: 18669667
If you know of a relevant reference for Tertiapin LQ, please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: Tertiapin LQ, Tertiapin LQ supplier, TertiapinLQ, kir1.1, blockers, selective, venoms, inward, rectifier, potassium, channels, Inward, Potassium, Channels, 4339, Tocris Bioscience
Citations for Tertiapin LQ
Citations are publications that use Tocris products.
Currently there are no citations for Tertiapin LQ. Do you know of a great paper that uses Tertiapin LQ from Tocris? Please let us know.
Reviews for Tertiapin LQ
There are currently no reviews for this product. Be the first to review Tertiapin LQ and earn rewards!
Have you used Tertiapin LQ?
Submit a review and receive an Amazon gift card.
$50/€35/£30/$50CAN/¥300 Yuan/¥5000 Yen for first to review with an image
$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image
Literature in this Area
Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!
*Please note that Tocris will only send literature to established scientific business / institute addresses.
Cardiovascular Research Product Guide
A collection of over 250 products for cardiovascular research, the guide includes research tools for the study of:
- Hypertension
- Thrombosis and Hemostasis
- Atherosclerosis
- Myocardial Infarction
- Ischemia/Reperfusion Injury
- Arrhythmias
- Heart Failure
Ion Channel Product Listing
A collection of around 500 products for ion channel research, the listing includes research tools for the study of:
- Ligand-gated ion channels
- Voltage-gated ion channels
- Other Ion Channels
Pain Research Product Guide
A collection of over 280 products for pain research, the guide includes research tools for the study of:
- Nociception
- Ion Channels
- G-Protein-Coupled Receptors
- Intracellular Signaling