MR 16728 hydrochloride

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Cat.No. 0537 - MR 16728 hydrochloride | C23H36N2O.HCl | CAS No. 207403-36-9
Description: Stimulates ACh release
Chemical Name: N-[3-(1-Hexahydroazapinyl)propyl]-α-cyclohexyl-benzeneacetamide hydrochloride
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Biological Activity

This analog of cetiedil stimulates the release of acetylcholine from synaptosomes.

Technical Data

M. Wt 393.01
Formula C23H36N2O.HCl
Storage Desiccate at -20°C
CAS Number 207403-36-9
PubChem ID 378810
InChI Key QLMQSFIGPVLVAO-UHFFFAOYSA-N
Smiles Cl.O=C(NCCCN1CCCCCC1)C(C1CCCCC1)C1=CC=CC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Solubility Data

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 39.3 100

Preparing Stock Solutions

The following data is based on the product molecular weight 393.01. Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.54 mL 12.72 mL 25.44 mL
5 mM 0.51 mL 2.54 mL 5.09 mL
10 mM 0.25 mL 1.27 mL 2.54 mL
50 mM 0.05 mL 0.25 mL 0.51 mL

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References

References are publications that support the biological activity of the product.

Moulian et al (1993) The effect of MR 16728, a cetiedil analogue, on acetylcholine release in torpedo synaptosomes. Eur.J.Pharmacol. 231 407 PMID: 8449232


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Citations for MR 16728 hydrochloride

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