MCOPPB trihydrochloride

Discontinued Product

MCOPPB trihydrochloride (Cat. No. 3763) has been withdrawn from sale for commercial reasons.
Description: Potent NOP receptor agonist
Chemical Name: 1-[1-(1-Methylcyclooctyl)-4-piperidinyl]-2-(3R)-3-piperidinyl-1H-benzimidazole trihydrochloride
Purity: ≥99% (HPLC)
Literature (1)

Biological Activity for MCOPPB trihydrochloride

MCOPPB trihydrochloride is a high affinity NOP receptor agonist (pKi = 10.07 for the human NOP receptor). Exhibits anxiolytic effects with no effect on memory or locomotion. Regarded as one of the most potent, non-peptide NOP full agonists in vitro.

Licensing Information

Sold for research purposes under agreement from Pfizer Inc.

Technical Data for MCOPPB trihydrochloride

M. Wt 534.05
Formula C26H40N4.3HCl
Storage Store at -20°C
Purity ≥99% (HPLC)
CAS Number 1108147-88-1
PubChem ID 25208093
Smiles CC5(CCCCCCC5)N(CC4)CCC4N2C1=CC=CC=C1N=[C@@]2[C@H]3CNCCC3.Cl.Cl.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for MCOPPB trihydrochloride

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Citations for MCOPPB trihydrochloride

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Currently there are no citations for MCOPPB trihydrochloride.

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

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Peptides Involved in Appetite Modulation Scientific Review

Peptides Involved in Appetite Modulation Scientific Review

Written by Sonia Tucci, Lynsay Kobelis and Tim Kirkham, this review provides a synopsis of the increasing number of peptides that have been implicated in appetite regulation and energy homeostasis; putative roles of the major peptides are outlined and compounds available from Tocris are listed.