HomoAMPA
Discontinued Product
Unfortunately HomoAMPA (Cat. No. 1026) has been withdrawn from sale for commercial reasons.
Biological Activity
The higher homolog of AMPA, this compound is completely inactive at ionotropic glutamate receptors but instead is a relatively potent and highly mGlu6 subtype-selective metabotropic glutamate receptor agonist.
Technical Data
| M. Wt | 200.19 |
| Formula | C8H12N2O4 |
| Storage | Store at RT |
| Smiles | Cc1c(CCC(C(=O)O)N)c(no1)O |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Preparing Stock Solutions
The following data is based on the product molecular weight 200.19. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 5 mL | 24.98 mL | 49.95 mL |
| 5 mM | 1 mL | 5 mL | 9.99 mL |
| 10 mM | 0.5 mL | 2.5 mL | 5 mL |
| 50 mM | 0.1 mL | 0.5 mL | 1 mL |
Molarity Calculator
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Product Datasheets
References
References are publications that support the products' biological activity.
Brauner-Osbourne et al (1996) A new highly selective metabotropic excitatory amino acid agonist: 2-amino-4-(3-hydroxy-5-methylisoxazole-4-yl)butyric acid. J.Med.Chem. 39 3188 PMID: 8759641
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Keywords: HomoAMPA, supplier, Potent, selective, mGlu6, agonists, mGlur, Group, III, Receptors, mGluR6, Glutamate, Metabotropic, Glutamate, (Metabotropic), Group, III, Receptors, Tocris Bioscience
Citations for HomoAMPA
Citations are publications that use Tocris products.
Currently there are no citations for HomoAMPA.
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