(±)-ACPT-III

Discontinued Product

(±)-ACPT-III (Cat. No. 1113) has been withdrawn from sale for commercial reasons.
Cat.No. 1113 - (±)-ACPT-III | C8H11NO6
Description: Selective group III agonist
Chemical Name: (3RS,4RS)-1-Aminocyclopentane-1,3,4-tricarboxylic acid
Datasheet
Citations
Reviews
Literature

Biological Activity

A selective group III metabotropic receptor agonist displaying EC50 values of 40 μM at mGlu4a receptors and > 1 mM at mGlu1a and mGlu2 receptors.

Licensing Information

Sold with the permission of the CNRS.

Technical Data

M. Wt 217.18
Formula C8H11NO6
Storage Desiccate at -20°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

References

References are publications that support the biological activity of the product.

Acher et al (1997) Synthesis and pharmacological characterization of aminocyclopentanetricarboxylic acids: new tools to discriminate between metabotropic glutamate receptor.subtypes J.Med.Chem. 40 3119 PMID: 9301676

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Keywords: (±)-ACPT-III, (±)-ACPT-III supplier, Glutamate, (Metabotropic), Group, III, Receptors, 1113, Tocris Bioscience

Citations for (±)-ACPT-III

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Currently there are no citations for (±)-ACPT-III.

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Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* or download your copy today!

*Please note that Tocris will only send literature to established scientific business / institute addresses.


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