Desloratadine

Discontinued Product

Desloratadine (Cat. No. 5958) has been withdrawn from sale for commercial reasons.
Cat.No. 5958 - Desloratadine | C19H19ClN2 | CAS No. 100643-71-8
Description: High affinity H1 antagonist; anti-inflammatory
Chemical Name: 8-Chloro-6,11-dihydro-11-(4-piperidinylidene)-5H-benzo[5,6]cyclohepta[1,2-b]pyridine
Purity: ≥99% (HPLC)
Datasheet
Citations
Reviews
Literature (3)

Biological Activity for Desloratadine

Desloratadine is a high affinity histamine H1 receptor antagonist (Ki = 0.87 nM); active metabolite of loratadine (Cat. No. 1944). Anti-inflammatory.

Technical Data for Desloratadine

M. Wt 310.82
Formula C19H19ClN2
Storage Store at +4°C
Purity ≥99% (HPLC)
CAS Number 100643-71-8
PubChem ID 124087
InChI Key JAUOIFJMECXRGI-UHFFFAOYSA-N
Smiles ClC1=CC=C2C(CCC3=C(/C2=C4CCNCC\4)N=CC=C3)=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for Desloratadine

References for Desloratadine

References are publications that support the biological activity of the product.

Henz (2001) The pharmacologic profile of desloratadine: a review. Allergy 56 7 PMID: 11243504

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Citations for Desloratadine

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Currently there are no citations for Desloratadine.

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