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Cat.No. 0543 - C-1 | C13H15N3O2S | CAS No. 84468-24-6
Description: Protein kinase C inhibitor
Chemical Name: 1-(5-Isoquinolinesulfonyl)piperazine
Purity: ≥99% (HPLC)

Biological Activity

Inhibitor of protein kinase C. Vasodilator.

Compound Libraries

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Technical Data

M. Wt 277.34
Formula C13H15N3O2S
Storage Store at RT
Purity ≥99% (HPLC)
CAS Number 84468-24-6
PubChem ID 3545
Smiles O=S(=O)(N1CCNCC1)C1=C2C=CN=CC2=CC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solvent Max Conc. mg/mL Max Conc. mM
DMSO 27.73 100

Preparing Stock Solutions

The following data is based on the product molecular weight 277.34. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.61 mL 18.03 mL 36.06 mL
5 mM 0.72 mL 3.61 mL 7.21 mL
10 mM 0.36 mL 1.8 mL 3.61 mL
50 mM 0.07 mL 0.36 mL 0.72 mL

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Product Datasheets

Safety Datasheet


References are publications that support the products' biological activity.

Gerard et al (1986) Role of protein kinases in stimulation of human polymorphonuclear leukocyte oxidation metabolism by various agonists. J.Clin.Invest. 77 61 PMID: 3003155

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Keywords: C-1, supplier, Protein, kinase, C, inhibitors, inhibits, PKC, Kinases, vasodilator, Protein, Kinase, C, Protein, Kinase, C, Tocris Bioscience

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