BTCP maleate

Discontinued Product

Unfortunately BTCP maleate (Cat. No. 0702) has been withdrawn from sale for commercial reasons.
Cat.No. 0702 - BTCP maleate | C19H25NS.C4H4O4 | CAS No. 207455-25-2
Description: Potent dopamine uptake inhibitor
Chemical Name: 1-[1-(2-Benzo[b]thienyl)cyclohexyl)]piperidine maleate
Purity: ≥98% (HPLC)
Datasheet
Citations
Reviews
Literature

Biological Activity

A potent dopamine re-uptake inhibitor with a behavioral profile different from that of PCP and similar to that of cocaine.

Compound Libraries

BTCP maleate is also offered as part of the Tocriscreen Plus. Find out more about compound libraries available from Tocris.

Technical Data

M. Wt 415.55
Formula C19H25NS.C4H4O4
Storage Desiccate at +4°C
Purity ≥98% (HPLC)
CAS Number 207455-25-2
PubChem ID 10251290
InChI Key AMTYJSWZECGJOO-BTJKTKAUSA-N
Smiles OC(=O)\C=C/C(O)=O.C1CCN(CC1)C1(CCCCC1)C1=CC2=CC=CC=C2S1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Preparing Stock Solutions

The following data is based on the product molecular weight 415.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.41 mL 12.03 mL 24.06 mL
5 mM 0.48 mL 2.41 mL 4.81 mL
10 mM 0.24 mL 1.2 mL 2.41 mL
50 mM 0.05 mL 0.24 mL 0.48 mL

Molarity Calculator

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Reconstitution Calculator

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Product Datasheets

Safety Datasheet

References

References are publications that support the products' biological activity.

Chergui et al (1992) Inhibition of the locus coeruleus neurons by the phenylcyclidine analog, N-[1-(2-benzo(b thiophenyl)cyclohexyl]-piperidine: evidence for potent indirect adrenoceptor agonist properties. Eur.J.Pharmacol. 219 169 PMID: 1397045

Koek et al (1989) The phencyclidine (PCP) analogue N-[1-(2-benzo(b)thiophenyl)cyclohexyl]piperidine shares cocaine-like but not other characteristic behavioural effects with PCP, ketamine and MK-801. J.Pharmacol.Exp.Ther. 250 1019 PMID: 2674416

Vignon et al (1988) [3H]N-[1-(2-benzo[b]thiophenyl)cyclohexyl]piperidine ([3H]BTCP): a new phencyclidine analogue selective for the dopamine uptake complex. Eur.J.Pharmacol. 148 427 PMID: 3384005

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Keywords: BTCP maleate, supplier, Potent, dopamine, reuptake, inhibitors, inhibits, DAT, Transporters, Monoamine, Neurotransmitter, Dopamine, Transporters, Dopamine, Transporters, Tocris Bioscience

Citations for BTCP maleate

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