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Submit ReviewTC-P 262 is a selective P2X3 and P2X2/3 receptor antagonist (pIC50 values are 7.39 and 6.68 respectively). Displays no detectable activity at P2X1, P2X2, P2X4 and P2X7 receptors (pIC50 < 4.7).
M. Wt | 258.32 |
Formula | C14H18N4O |
Storage | Store at RT |
Purity | ≥99% (HPLC) |
CAS Number | 873398-67-5 |
PubChem ID | 59598765 |
InChI Key | RAKSAPLZNJXYRB-UHFFFAOYSA-N |
Smiles | NC1=NC(N)=NC=C1OC2=C(C(C)C)C=CC(C)=C2 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
References are publications that support the biological activity of the product.
Ballini et al (2011) Characterization of three diaminopyrimidines as potent and selective antagonists of P2X3 and P2X2/3 receptors with in vivo efficacy in a pain model. Br.J.Pharmacol. 163 1315 PMID: 21410458
Keywords: TC-P 262, TC-P 262 supplier, Selective, P2X3, P2X2/3, receptors, antagonists, TC-P262, P2X, Receptors, 4386, Tocris Bioscience
Citations are publications that use Tocris products. Selected citations for TC-P 262 include:
Hui et al (2020) Simultaneous Control of Endogenous and User-Defined Genetic Pathways Using Unique ecDHFR Pharmacological Chaperones. Cell Chem Biol 27 622-634.e6 PMID: 32330442
Average Rating: 4 (Based on 1 Review.)
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