Potent and selective adenosine A2B receptor antagonist (IC50 = 3.64 nM at human A2B receptors). Displays > 100-fold selectivity over hA1, hA2A and hA3 receptors.
|Storage||Store at +4°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
|Solvent||Max Conc. mg/mL||Max Conc. mM|
Preparing Stock Solutions
The following data is based on the product molecular weight 543.04. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.84 mL||9.21 mL||18.41 mL|
|5 mM||0.37 mL||1.84 mL||3.68 mL|
|10 mM||0.18 mL||0.92 mL||1.84 mL|
|50 mM||0.04 mL||0.18 mL||0.37 mL|
References are publications that support the products' biological activity.
Borrmann et al (2009) 1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity. J.Med.Chem. 52 3994 PMID: 19569717
If you know of a relevant reference for PSB 0788, please let us know.
View Related Products by Product Action
Keywords: PSB 0788, supplier, Selective, A2B, antagonists, Receptors, adenosines, PSB0788, Adenosine, A2B, Receptors, Adenosine, A2B, Receptors, Tocris Bioscience
Citations for PSB 0788
Citations are publications that use Tocris products.
Currently there are no citations for PSB 0788. Do you know of a great paper that uses PSB 0788 from Tocris? If so please let us know.
Reviews for PSB 0788
There are currently no reviews for this product. Be the first to review PSB 0788 and earn rewards!
Have you used PSB 0788?
Submit a review and receive an Amazon gift card.
$10US/$10CAN/€7/£6 gift card for a review without an image
$25US/$25CAN/€18/£15 gift card for a review with an image
*Offer only valid in the USA / Canada, UK and EuropeSubmit a Review