Discontinued Product

(-)-5'-DMH-CBD (Cat. No. 1481) has been withdrawn from sale for commercial reasons.
Description: Metabolically stable anandamide transport inhibitor
Alternative Names: (-)-5'-Dimethylheptyl-cannabidiol
Chemical Name: 5-(1,1-Dimethylheptyl)-2-[(1R,6R)-3-methyl-6-(1-methylethenyl)-2-cyclohexen-1-yl]-1,3-benzenediol
Literature (2)

Biological Activity for (-)-5'-DMH-CBD

(-)-5'-DMH-CBD is an anandamide membrane transport inhibitor (IC50 = 14 μM) that is relatively metabolically stable. Displays some affinity for CB2 receptors but has only weak affinity for CB1 receptors and has no activity at VR1 receptors or FAAH. Anticonvulsive in vivo following systemic administration.

Technical Data for (-)-5'-DMH-CBD

M. Wt 370.57
Formula C25H38O2
Storage Desiccate at -20°C
CAS Number 97452-63-6
PubChem ID 126670
Smiles C=[C@](C)[C@@H]1CCC(C)=C[C@H]1[C@]2=C(O)C=C(C(C)(C)CCCCCC)C=C2O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for (-)-5'-DMH-CBD

Certificate of Analysis / Product Datasheet
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References for (-)-5'-DMH-CBD

References are publications that support the biological activity of the product.

Bisogno et al (2001) Molecular targets for cannabidiol and its synthetic analogues: effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamide. Br.J.Pharmacol. 134 845 PMID: 11606325

Leite et al (1982) Anticonvulsant effects of the (-) and (+)isomers of cannabidiol and their dimethylheptyl homologs. Pharmacology 24 141 PMID: 7071126

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Citations for (-)-5'-DMH-CBD

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

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