(-)-5'-DMH-CBD

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Cat.No. 1481 - (-)-5'-DMH-CBD | C25H38O2 | CAS No. 97452-63-6
Description: Metabolically stable anandamide transport inhibitor
Alternative Names: (-)-5'-Dimethylheptyl-cannabidiol
Chemical Name: 5-(1,1-Dimethylheptyl)-2-[(1R,6R)-3-methyl-6-(1-methylethenyl)-2-cyclohexen-1-yl]-1,3-benzenediol
Datasheet
Citations
Reviews
Literature

Biological Activity

Anandamide membrane transport inhibitor (IC50 = 14 μM) that is relatively metabolically stable. Displays some affinity for CB2 receptors but has only weak affinity for CB1 receptors and has no activity at VR1 receptors or FAAH. Anticonvulsive in vivo following systemic administration.

Technical Data

M. Wt 370.57
Formula C25H38O2
Storage Desiccate at -20°C
CAS Number 97452-63-6
PubChem ID 126670
InChI Key MPJURNPNPDQYSY-LEWJYISDSA-N
Smiles C=[C@](C)[C@@H]1CCC(C)=C[C@H]1[C@]2=C(O)C=C(C(C)(C)CCCCCC)C=C2O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solubility Soluble in ethanol (supplied pre-dissolved in anhydrous ethanol, 5mg/ml)

Product Datasheets

Certificate of Analysis / Product Datasheet
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References

References are publications that support the biological activity of the product.

Bisogno et al (2001) Molecular targets for cannabidiol and its synthetic analogues: effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamide. Br.J.Pharmacol. 134 845 PMID: 11606325

Leite et al (1982) Anticonvulsant effects of the (-) and (+)isomers of cannabidiol and their dimethylheptyl homologs. Pharmacology 24 141 PMID: 7071126


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Citations for (-)-5'-DMH-CBD

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Literature in this Area

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