Methyl 2,5-dihydroxycinnamate

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Cat.No. 0577 - Methyl 2,5-dihydroxycinnamate | C10H10O4 | CAS No. 63177-57-1
Description: EGFR-kinase inhibitor
Alternative Names: Erbstatin analog
Purity: ≥98% (HPLC)
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Biological Activity

Erbstatin analog. Inhibitor of EGF receptor-associated tyrosine kinases.

Technical Data

M. Wt 194.19
Formula C10H10O4
Storage Store at RT
Purity ≥98% (HPLC)
CAS Number 63177-57-1
PubChem ID 5353609
InChI Key BQCNSTFWSKOWMA-GORDUTHDSA-N
Smiles COC(=O)\C=C\C1=C(O)C=CC(O)=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

SolubilitySoluble to 100 mM in ethanol

Preparing Stock Solutions

The following data is based on the product molecular weight 194.19. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 5.15 mL 25.75 mL 51.5 mL
5 mM 1.03 mL 5.15 mL 10.3 mL
10 mM 0.51 mL 2.57 mL 5.15 mL
50 mM 0.1 mL 0.51 mL 1.03 mL

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Product Datasheets

Safety Datasheet

References

References are publications that support the products' biological activity.

Isshiki et al (1990) Inhibition of epidermal growth factor-induced DNA synthesis by tyrosine kinase inhibitors. FEBS Lett. 260 198 PMID: 2298299


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Citations for Methyl 2,5-dihydroxycinnamate

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