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Centrally active opioid analgesic. Partial agonist at the μ1 opioid receptor. Also shown to inhibit acetylcholinesterase.
|Storage||Desiccate at +4°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
|Solvent||Max Conc. mg/mL||Max Conc. mM|
Preparing Stock Solutions
The following data is based on the product molecular weight 269.81. Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||3.71 mL||18.53 mL||37.06 mL|
|5 mM||0.74 mL||3.71 mL||7.41 mL|
|10 mM||0.37 mL||1.85 mL||3.71 mL|
|50 mM||0.07 mL||0.37 mL||0.74 mL|
References are publications that support the biological activity of the product.
Spiegel and Pasternak (1984) Meptazinol: a novel Mu-1 selective opioid analgesic. J.Pharmacol.Exp.Ther. 228 414 PMID: 6141283
Galli et al (1996) Reversible inhibition of cholinesterases by opioids: possible pharmacological consequences. J.Pharm.Pharmacol. 48 116
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Keywords: Meptazinol hydrochloride, Meptazinol hydrochloride supplier, Partial, agonists, μ1-opioid, mu1-opioid, Receptors, MOP, OP3, μ-opioid, mu-opioid, Mu, Opioid, 3636, Tocris Bioscience
Citations for Meptazinol hydrochloride
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Literature in this Area
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