Selective δ opioid antagonist.
Sold with the permission of AstraZeneca UK Ltd.
(Modifications: Tyr-1 = N,N-diallyl-Tyr, Gly-2 - Phe-3 peptide bond replaced with Psi-(CH2S))
|Storage||Desiccate at -20°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
|Solubility||Soluble to 1 mg/ml in methanol|
Preparing Stock Solutions
The following data is based on the product molecular weight 638.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.57 mL||7.83 mL||15.65 mL|
|5 mM||0.31 mL||1.57 mL||3.13 mL|
|10 mM||0.16 mL||0.78 mL||1.57 mL|
|50 mM||0.03 mL||0.16 mL||0.31 mL|
References are publications that support the products' biological activity.
Shaw et al (1982) Selective antagonists at the opiate delta-receptor. Life Sci. 31 1259 PMID: 6128652
If you know of a relevant reference for ICI 154,129, please let us know.
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Keywords: ICI 154,129, supplier, δ-opioid, delta-opioid, selective, peptide, antagonists, DOP, Receptors, OP1, ICI154129, AstraZeneca, Delta, Opioid, Receptors, Delta, Opioid, Receptors, Tocris Bioscience
1 Citation for ICI 154,129
Citations are publications that use Tocris products. Selected citations for ICI 154,129 include:
Jiang et al (2015) Analgesic roles of peripheral intrinsic met-enkephalin and dynorphin A in long-lasting inflammatory pain induced by complete Freund's adjuvant in rats. J Pharmacol Exp Ther 9 2344 PMID: 26136984
Do you know of a great paper that uses ICI 154,129 from Tocris? If so please let us know.
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