Etonitazenyl isothiocyanate

Discontinued Product

Unfortunately Etonitazenyl isothiocyanate (Cat. No. 0516) has been withdrawn from sale for commercial reasons.
Cat.No. 0516 - Etonitazenyl isothiocyanate | C23H28N4OS | CAS No. 85951-65-1
Description: Irreversible affinity label (μ selective)
Alternative Names: BIT
Chemical Name: 2-[(4-Ethoxyphenyl)methyl]-N,N-diethyl-5-isothiocyano-1H-benzimidazole-1-ethanamine

Biological Activity

Affinity label specific for μ opioid sites.

Technical Data

M. Wt 408.56
Formula C23H28N4OS
Storage Desiccate at -20°C
CAS Number 85951-65-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Preparing Stock Solutions

The following data is based on the product molecular weight 408.56. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.45 mL 12.24 mL 24.48 mL
5 mM 0.49 mL 2.45 mL 4.9 mL
10 mM 0.24 mL 1.22 mL 2.45 mL
50 mM 0.05 mL 0.24 mL 0.49 mL

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Product Datasheets

Certificate of Analysis is currently unavailable
on-line. Please contact Customer Service.
Safety Datasheet


References are publications that support the products' biological activity.

Burke et al (1984) Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for μ or δ opiate receptors. J.Med.Chem. 27 1570 PMID: 6150112

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Keywords: Irreversible affinity label μ-opioid mu-opioid selective MOP Receptors OP3 BIT Mu Opioid Receptors

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