Etonitazenyl isothiocyanate

Cat. No. 0516 Datasheet / COA / SDS

Discontinued Product

Unfortunately Etonitazenyl isothiocyanate (Cat. No. 0516) has been withdrawn from sale for commercial reasons.
Cat.No. 0516 - Etonitazenyl isothiocyanate | C23H28N4OS | CAS No. 85951-65-1
Description: Irreversible affinity label (μ selective)
Alternative Names: BIT
Chemical Name: 2-[(4-Ethoxyphenyl)methyl]-N,N-diethyl-5-isothiocyano-1H-benzimidazole-1-ethanamine
Datasheet
Citations
Reviews
Literature

Biological Activity

Affinity label specific for μ opioid sites.

Technical Data

M. Wt 408.56
Formula C23H28N4OS
Storage Desiccate at -20°C
CAS Number 85951-65-1
Smiles N#CSC1=CC=C2C(N=C(CC3=CC=C(OCC)C=C3)N2CCN(CC)CC)=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Product Datasheets

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Safety Datasheet

References

References are publications that support the products' biological activity.

Burke et al (1984) Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for μ or δ opiate receptors. J.Med.Chem. 27 1570 PMID: 6150112

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Citations for Etonitazenyl isothiocyanate

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