Potent δ-opioid receptor agonist (IC50 = 0.5 nM in human granulocytes). Exhibits a high rate of blood-brain barrier penetrance.
(Modifications: Ala-2 = D-Ala, Gly-7 = C-terminal amide)
|Storage||Store at -20°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
|Solubility||Soluble to 0.40 mg/ml in 50% acetonitrile / water|
Preparing Stock Solutions
The following data is based on the product molecular weight 768.87. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.3 mL||6.5 mL||13.01 mL|
|5 mM||0.26 mL||1.3 mL||2.6 mL|
|10 mM||0.13 mL||0.65 mL||1.3 mL|
|50 mM||0.03 mL||0.13 mL||0.26 mL|
The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.
References are publications that support the products' biological activity.
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Keywords: DeltorphinI delta d δ opioids agonists brain penetrant bbb Delta Opioid Receptors
1 Citation for Deltorphin I
Citations are publications that use Tocris products. Selected citations for Deltorphin I include:
Otis et al (2011) Spinal activation of delta opioid receptors alleviates cancer-related bone pain. Neuroscience 183 221 PMID: 21458544
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Literature in this Area
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