BP 554 maleate

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Cat.No. 0556 - BP 554 maleate | C20H24N2O3.C4H4O4 | CAS No. 1221401-95-1
Description: Selective 5-HT1A agonist
Chemical Name: 1-[3-(3,4-Methylenedioxyphenoxy)propyl]-4-phenyl-piperazine maleate
Purity: ≥99% (HPLC)
Datasheet
Citations (1)
Literature

Biological Activity

Selective 5-HT1A agonist.

Compound Libraries

BP 554 maleate is also offered as part of the Tocriscreen Plus. Find out more about compound libraries available from Tocris.

Technical Data

M. Wt 456.48
Formula C20H24N2O3.C4H4O4
Storage Store at RT
Purity ≥99% (HPLC)
CAS Number 1221401-95-1
PubChem ID 56972150
InChI Key NBCXNOHQTALBRA-BTJKTKAUSA-N
Smiles OC(=O)\C=C/C(O)=O.C(COC1=CC=C2OCOC2=C1)CN1CCN(CC1)C1=CC=CC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 45.65 100

Preparing Stock Solutions

The following data is based on the product molecular weight 456.48. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.19 mL 10.95 mL 21.91 mL
5 mM 0.44 mL 2.19 mL 4.38 mL
10 mM 0.22 mL 1.1 mL 2.19 mL
50 mM 0.04 mL 0.22 mL 0.44 mL

Molarity Calculator

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Reconstitution Calculator

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Dilution Calculator

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Product Datasheets

Safety Datasheet

References

References are publications that support the products' biological activity.

Matsuda et al (1989) Agonist activity of a novel compound, 1-[3-(3,4-methylenedioxyphenoxy)propyl]-4-phenyl piperazine (BP-554) at central 5-HT1A receptors. Eur.J.Pharmacol. 170 75 PMID: 2533078


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View all 5-HT1A Receptor Agonists

Keywords: Selective 5-HT1A agonists Serotonin Receptors 5-HT1 BP554 maleate 5-HT1A Receptors

1 Citation for BP 554 maleate

Citations are publications that use Tocris products. Selected citations for BP 554 maleate include:

Huang et al (2009) Autocrine and paracrine roles for ATP and serotonin in mouse taste buds. Br J Pharmacol 29 13909 PMID: 19890001


Do you know of a great paper that uses BP 554 maleate from Tocris? If so please let us know.

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Reviews

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Pathways for BP 554 maleate

Protocols

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