Arecaidine propargyl ester tosylate

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Cat.No. 0383 - Arecaidine propargyl ester tosylate | C10H13NO2.C7H8SO3 | CAS No. 147202-94-6
Description: Muscarinic agonist
Chemical Name: N-Methyl-1,2,5,6-tetrahydropyridine-3-carboxylic acid propargyl ester tosylate
Datasheet
Citations
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Literature

Biological Activity

A potent muscarinic receptor agonist. Shows some selectivity for cardiac versus ileal M2 receptors.

Technical Data

M. Wt 351.42
Formula C10H13NO2.C7H8SO3
Storage Store at RT
CAS Number 147202-94-6
PubChem ID 6604936
InChI Key LYHWIOMAWPVTPI-UHFFFAOYSA-N
Smiles CC1=CC=C(C=C1)S(O)(=O)=O.CN1CCC=C(C1)C(=O)OCC#C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Solubility Data

Solubility Soluble to 100 mM in water

References

References are publications that support the biological activity of the product.

Barlow and Weston-Smith (1985) The relative potencies of some agonists at M2 muscarinic receptors in guinea pig ileum, atria and bronchi. Br.J.Pharmacol. 85 437 PMID: 3896364

Moser et al (1989) Structure-activity relationships of new analogues of arecaidine propargyl ester at muscarinic M1 and M2 receptor subtypes. Br.J.Pharmacol. 96 319 PMID: 2924082


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Keywords: Arecaidine propargyl ester tosylate, Arecaidine propargyl ester tosylate supplier, Muscarinic, agonists, Receptors, Acetylcholine, Ach, M2, 0383, Tocris Bioscience

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