Discontinued Product

6,2',4'-Trimethoxyflavone (Cat. No. 3859) has been withdrawn from sale for commercial reasons.
Cat.No. 3859 - 6,2',4'-Trimethoxyflavone | C18H16O5 | CAS No. 720675-74-1
Description: Aryl hydrocarbon receptor antagonist
Chemical Name: 2',4',6-Trimethoxyflavone
Purity: ≥97% (HPLC)
Citations (1)
Reviews (1)
Literature (1)

Biological Activity for 6,2',4'-Trimethoxyflavone

6,2',4'-Trimethoxyflavone is an aryl hydrocarbon receptor antagonist (EC50 = 0.9 μM). Exhibits no short term agonist activity and no species or promoter dependence.

Technical Data for 6,2',4'-Trimethoxyflavone

M. Wt 312.32
Formula C18H16O5
Storage Store at RT
Purity ≥97% (HPLC)
CAS Number 720675-74-1
PubChem ID 688802
Smiles O=C1C3=C(C=CC(OC)=C3)OC(C2=CC=C(OC)C=C2OC)=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for 6,2',4'-Trimethoxyflavone

Certificate of Analysis / Product Datasheet
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References for 6,2',4'-Trimethoxyflavone

References are publications that support the biological activity of the product.

Murray et al (2010) Antagonism of aryl hydrocarbon receptor signaling by 6,2',4'-trimethoxyflavone. J.Pharmacol.Exp.Ther. 332 135 PMID: 19828881

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Keywords: 6,2',4'-Trimethoxyflavone, 6,2',4'-Trimethoxyflavone supplier, aryl, hydrocarbon, receptors, antagonists, AHR, 6,2,4-Trimethoxyflavone, Aryl, Hydrocarbon, Receptors, 3859, Tocris Bioscience

1 Citation for 6,2',4'-Trimethoxyflavone

Citations are publications that use Tocris products. Selected citations for 6,2',4'-Trimethoxyflavone include:

Gimenez-Gomez et al (2018) Increasing kynurenine brain levels reduces ethanol consumption in mice by inhibiting dopamine release in nucleus accumbens. Neuropharmacology 135 581 PMID: 29705534

Reviews for 6,2',4'-Trimethoxyflavone

Average Rating: 5 (Based on 1 Review.)

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Good choice.
By Anonymous on 08/20/2018
Assay Type: In Vitro
Species: Human

Purchased to independently test published results and was successful. Compound purity was as described. Happy with purchase

Literature in this Area

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