Cat. No. 2974
Chemical Name: 3-Methyl-3-propyl-1,1,2,2-cycloprop
Biological ActivityInhibitor of regulator of G-protein signaling 4 (RGS4). Reduces the RGS4-Gαo protein-protein interaction signal.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
Roman et al (2007) Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay. Mol.Pharmacol. 71 169. PMID: 17012620.
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Citations are publications that use Tocris products. Selected citations for CCG 2046 include:
Leister et al (2011) Two High Throughput Screen Assays for Measurement of TNF-α in THP-1 Cells. Curr Chem Genomics 5 21. PMID: 21643507.
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Keywords: CCG 2046, supplier, inhibitors, inhibits, regulator, G-protein, signaling, 4, RGS4, Gao, Heterotrimeric, CCG2046, Tocris Bioscience, G Protein (Heterotrimeric) Inhibitor products
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