TRPV Channel Antagonists
| Cat. No. | 产品名称/活性 |
|---|---|
| 5781 | A 425619 |
| Potent TRPV1 antagonist | |
| 4319 | A 784168 |
| Potent and selective TRPV1 antagonist | |
| 4330 | AMG 21629 |
| Potent and selective TRPV1 antagonist | |
| 5995 | AMG 517 |
| Potent TRPV1 antagonist | |
| 2316 | AMG 9810 |
| Potent and selective TRPV1 competitive antagonist | |
| 3875 | BCTC |
| TRPV1 antagonist | |
| 0464 | Capsazepine |
| TRPV antagonist; also activator of ENaCδ | |
| 5106 | GSK 2193874 |
| Potent and selective TRPV4 antagonist; orally active | |
| 4100 | HC 067047 |
| Potent and selective TRPV4 antagonist | |
| 3361 | JNJ 17203212 |
| Reversible, competitive and potent TRPV1 antagonist | |
| 3746 | RN 1734 |
| Selective TRPV4 antagonist | |
| 5678 | RN 9893 hydrochloride |
| Potent and selective TRPV4 antagonist | |
| 1439 | Ruthenium Red |
| Blocks capsaicin-activated cation channels | |
| 1615 | SB 366791 |
| Potent and selective TRPV1 competitive antagonist | |
| 6990 | SET 2 |
| Selective TRPV2 antagonist | |
| 1098 | Tranilast |
| Antiallergic; inhibits TRPV2-mediated responses | |
| 6831 | TRPV3 74a |
| Selective TRPV3 antagonist; brain penetrant |