Cat. No. |
产品名称/活性 |
5079 |
ABT 089 dihydrochloride |
| High affinity and selective α4β2 nAChR partial agonist |
6576 |
ABT 594 hydrochloride |
| Selective α4β2 nAChR agonist |
3549 |
3-Bromocytisine |
| Potent α4β4, α4β2 and α7 nAChR agonist |
5236 |
CC4 |
| High affinity and subtype-selective α6β2 and α4β2 nAChR partial agonist |
3546 |
(-)-Nicotine ditartrate |
| Prototypical nAChR agonist |
1053 |
RJR 2403 oxalate |
| Selective α4β2 nAChR agonist |
2737 |
TC 2559 difumarate |
| Selective α4β2 nAChR partial agonist |
6865 |
uPSEM 792 hydrochloride |
| α4β2 partial agonist; uPSEM agonist for PSAM4-GlyR and PSAM4-5HT3; brain-penetrant |
3754 |
Varenicline tartrate |
| Selective α4β2 nAChR partial agonist; orally active |