Discontinued Product

Sulfisoxazole (Cat. No. 0731) has been withdrawn from sale for commercial reasons.
Cat.No. 0731 - Sulfisoxazole | C11H13N3O3S | CAS No. 127-69-5
Description: Endothelin ETA antagonist
Chemical Name: 4-Amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide
Purity: ≥99% (HPLC)
Literature (5)

Biological Activity for Sulfisoxazole

Sulfisoxazole is a selective ETA endothelin receptor antagonist (IC50 values are 600 and 2200 nM for ETA and ETB receptors respectively).

Technical Data for Sulfisoxazole

M. Wt 267.3
Formula C11H13N3O3S
Storage Store at RT
Purity ≥99% (HPLC)
CAS Number 127-69-5
PubChem ID 5344
Smiles CC1=NOC(NS(=O)(=O)C2=CC=C(N)C=C2)=C1C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for Sulfisoxazole

References for Sulfisoxazole

References are publications that support the biological activity of the product.

Chan et al (1994) Identification of a new class of ETA selective endothelin antagonists by pharmacophore directed screening. Biochem.Biophys.Res.Commun. 201 228 PMID: 8198578

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Keywords: Sulfisoxazole, Sulfisoxazole supplier, Endothelin, ETA, antagonists, Receptors, 0731, Tocris Bioscience

Citations for Sulfisoxazole

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Currently there are no citations for Sulfisoxazole.

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Literature in this Area

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