PSB 603 - Bogus

Discontinued Product

PSB 603 - Bogus (Cat. No. 2683) has been withdrawn from sale for commercial reasons.
Cat.No. 2683 - PSB 603 | C24H25ClN6O4S
Description: Extremely selective A2B antagonist
Chemical Name: 8-[4-[4-(4-Chlorobenzyl)piperazide-1-sulfonyl)phenyl]]-1-propylxanthine
Purity: ≥98% (HPLC)
Datasheet
Citations
Reviews
Literature

Biological Activity

Adenosine A2B receptor antagonist that displays > 17000-fold selectivity over other adenosine receptors (Ki values are 0.568, > 10000, > 10000 and > 10000 nM for A2B, A1, A2A and A3 receptors respectively).

Technical Data

M. Wt 529.01
Formula C24H25ClN6O4S
Storage Store at +4°C
Purity ≥98% (HPLC)
Smiles O=C(NC2=C1NC(C3=CC=C(S(N4CCN(CC5=CC=C(Cl)C=C5)CC4)(=O)=O)C=C3)=N2)N(CCC)C1=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Product Datasheets

Certificate of Analysis is currently unavailable on-line.
Please contact Customer Service
Safety Datasheet

References

References are publications that support the biological activity of the product.

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Keywords: PSB 603, PSB 603 supplier, A2B, adenosine, Adenosine, Receptors, 2683, Tocris Bioscience

Citations for PSB 603 - Bogus

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* or download your copy today!

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Cardiovascular

Cardiovascular Poster

Cardiovascular disease remains one of the major causes of morbidity and mortality in the Western world and therefore this therapeutic area continues to be of great interest to researchers. This poster highlights the key GPCRs regulating vascular reactivity.