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Discontinued ProductMethimepip dihydrobromide (Cat. No. 2947) has been withdrawn from sale for commercial reasons.
Biological Activity for Methimepip dihydrobromide
Extremely selective histamine H3 receptor agonist (pKi values are 9.0, 5.7, < 5.0 and < 5.0 for hH3, hH4, hH1 and hH2 receptors respectively). Potently inhibits EFS-evoked contractions of guinea pig ileum (pD2 = 8.26).
Technical Data for Methimepip dihydrobromide
|Storage||Desiccate at RT|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for Methimepip dihydrobromide
References for Methimepip dihydrobromide
References are publications that support the biological activity of the product.
Kitbunnadaj et al (2005) N-substituted piperidinyl alkyl imidazoles: discovery of methimepip as a potent and selective histamine H3 receptor agonist. J.Med.Chem. 48 2100 PMID: 15771452
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Keywords: Methimepip dihydrobromide, Methimepip dihydrobromide supplier, selective, H3, agonists, Receptors, Histamine, histaminergic, 2947, Tocris Bioscience
Citations for Methimepip dihydrobromide
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Currently there are no citations for Methimepip dihydrobromide.
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Literature in this Area
Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!
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Alzheimer's disease (AD) is a degenerative brain disease and the most common cause of dementia, affecting approximately 47 million people worldwide. Updated in 2015, this poster summarizes the structural and functional changes observed in the progression of this neurodegenerative disease, as well as classic AD drug targets.