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Biological Activity for MA 2029
MA 2029 is a potent and selective, competitive motilin receptor antagonist (IC50 = 4.9 nM). Selective for the motilin receptor over a range of other receptors and ion channels. Inhibits motilin-induced duodenal muscle contractions in vitro. Also inhibits motilin-induced colonic and abdominal contractions in vivo. Orally active.
Technical Data for MA 2029
|Storage||Store at +4°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Solubility Data for MA 2029
|Solvent||Max Conc. mg/mL||Max Conc. mM|
Preparing Stock Solutions for MA 2029
The following data is based on the product molecular weight 556.71. Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.8 mL||8.98 mL||17.96 mL|
|5 mM||0.36 mL||1.8 mL||3.59 mL|
|10 mM||0.18 mL||0.9 mL||1.8 mL|
|50 mM||0.04 mL||0.18 mL||0.36 mL|
References for MA 2029
References are publications that support the biological activity of the product.
Sudo et al (2008) Oral administration of MA-2029, a novel selective and competitive motilin receptor antagonist, inhibits motilin-induced intestinal contractions and visceral pain in rabbits. Eur.J.Pharmacol. 581 296 PMID: 18164286
If you know of a relevant reference for MA 2029, please let us know.
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Keywords: MA 2029, MA 2029 supplier, MA2029, potent, selective, competitive, motilin, receptors, antagonists, Motilin, Receptors, 4934, Tocris Bioscience
Citations for MA 2029
Citations are publications that use Tocris products.
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Literature in this Area
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