ETB endothelin receptor antagonist.
(Modifications: Disulfide bridge between 1 - 5)
|Storage||Desiccate at -20°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
|Solubility||Soluble to 1 mg/ml in 20% acetonitrile|
Preparing Stock Solutions
The following data is based on the product molecular weight 1410. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||0.71 mL||3.55 mL||7.09 mL|
|5 mM||0.14 mL||0.71 mL||1.42 mL|
|10 mM||0.07 mL||0.35 mL||0.71 mL|
|50 mM||0.01 mL||0.07 mL||0.14 mL|
References are publications that support the biological activity of the product.
Haynes et al (1993) Endothelin; progress in pharmacology and physiology. TiPS 14 225 PMID: 8372400
Karaki et al (1993) ETB receptor antagonist, IRL 1038, selectively inhibits the endothelin-induced endothelium-dependent vascular relaxation. Eur.J.Pharmacol. 231 371 PMID: 8449230
If you know of a relevant reference for IRL-1038, please let us know.
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Keywords: IRL-1038, IRL-1038 supplier, ETB, antagonists, Receptors, Endothelin, 1195, Tocris Bioscience
1 Citation for IRL-1038
Citations are publications that use Tocris products. Selected citations for IRL-1038 include:
Khan et al (2006) Pharmacological characterization of endothelin receptors-mediated contraction in the mouse isolated proximal and distal colon. Br J Pharmacol 147 607 PMID: 16432510
Do you know of a great paper that uses IRL-1038 from Tocris? Please let us know.
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