Burimamide oxalate

Discontinued Product

Unfortunately Burimamide oxalate (Cat. No. 1857) has been withdrawn from sale for commercial reasons.
Cat.No. 1857 - Burimamide oxalate | C9H16N4S.C2H2O4 | CAS No. 163932-06-7
Description: Mixed H2/H3 antagonist
Chemical Name: N-[4-(1H-Imidazol-4-yl)butyl]-N'-methylthiourea oxalate

Biological Activity

Histamine H3/H2 receptor antagonist (Ki values are 0.07, 7.8 and 290 μM for H3, H2 and H1 receptors respectively). Displays partial agonist activity in SK-N-MC cells. Produces antinociceptive effects following intraventricular administration (ED50 = 183 nmol/mouse in hot-plate test).

Technical Data

M. Wt 302.35
Formula C9H16N4S.C2H2O4
Storage Desiccate at +4°C
CAS Number 163932-06-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Preparing Stock Solutions

The following data is based on the product molecular weight 302.35. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.31 mL 16.54 mL 33.07 mL
5 mM 0.66 mL 3.31 mL 6.61 mL
10 mM 0.33 mL 1.65 mL 3.31 mL
50 mM 0.07 mL 0.33 mL 0.66 mL

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Product Datasheets

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References are publications that support the products' biological activity.

Lamberti et al (1996) Investigation into the role of histamine receptors in rodent antinociception. Pharmacol.Biochem.Behav. 53 567 PMID: 8866956

Hough et al (2000) Antinociceptive activity of derivatives of improgran and burimamide. Pharmacol.Biochem.Behav. 65 61 PMID: 10638637

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Keywords: Burimamide oxalate, supplier, Mixed, H2/H3, antagonists, H3, Receptors, Histamine, H2, histaminergic, Histamine, H2, Receptors, Histamine, H3, Receptors, Histamine, H2, Receptors, Tocris Bioscience

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