Burimamide oxalate

Discontinued Product

Burimamide oxalate (Cat. No. 1857) has been withdrawn from sale for commercial reasons.
Description: Mixed H2/H3 antagonist
Chemical Name: N-[4-(1H-Imidazol-4-yl)butyl]-N'-methylthiourea oxalate
Literature (1)

Biological Activity for Burimamide oxalate

Histamine H3/H2 receptor antagonist (Ki values are 0.07, 7.8 and 290 μM for H3, H2 and H1 receptors respectively). Displays partial agonist activity in SK-N-MC cells. Produces antinociceptive effects following intraventricular administration (ED50 = 183 nmol/mouse in hot-plate test).

Technical Data for Burimamide oxalate

M. Wt 302.35
Formula C9H16N4S.C2H2O4
Storage Desiccate at +4°C
CAS Number 163932-06-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for Burimamide oxalate

References for Burimamide oxalate

References are publications that support the biological activity of the product.

Lamberti et al (1996) Investigation into the role of histamine receptors in rodent antinociception. Pharmacol.Biochem.Behav. 53 567 PMID: 8866956

Hough et al (2000) Antinociceptive activity of derivatives of improgran and burimamide. Pharmacol.Biochem.Behav. 65 61 PMID: 10638637

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Keywords: Burimamide oxalate, Burimamide oxalate supplier, Mixed, H2/H3, antagonists, H3, Receptors, Histamine, H2, histaminergic, 1857, Tocris Bioscience

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

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Histamine Receptors Scientific Review

Histamine Receptors Scientific Review

Written by Iwan de Esch and Rob Leurs, this review provides a synopsis of the different histamine receptor subtypes and the ligands that act upon them; compounds available from Tocris are listed.