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Submit ReviewArecaidine but-2-ynyl ester tosylate
Discontinued Product
Arecaidine but-2-ynyl ester tosylate (Cat. No. 0382) has been withdrawn from sale for commercial reasons.
Description: Muscarinic agonist
Chemical Name: N-Methyl-1,2,5,6-tetrahydropyridine-3-carboxylic acid but-2-ynyl ester tosylate
Biological Activity for Arecaidine but-2-ynyl ester tosylate
Potent muscarinic agonist, 4.6-fold selective for M2 receptors in the atrium versus those in the ileum.
Technical Data for Arecaidine but-2-ynyl ester tosylate
| M. Wt | 365.44 |
| Formula | C11H15NO2.C7H8SO3 |
| Storage | Store at RT |
| CAS Number | 119630-77-2 |
| Smiles | CC1=CC=C(C=C1)S(O)(=O)=O.CC#CCOC(=O)C1=CCCN(C)C1 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for Arecaidine but-2-ynyl ester tosylate
References for Arecaidine but-2-ynyl ester tosylate
References are publications that support the biological activity of the product.
Barlow and Weston-Smith (1985) The relative potencies of some agonists at M2 muscarinic receptors in guinea pig ileum, atria and bronchi. Br.J.Pharmacol. 85 437 PMID: 3896364
Moser et al (1989) Structure-activity relationships of new analogues of arecaidine propargyl ester at muscarinic M1 and M2 receptor subtypes. Br.J.Pharmacol. 96 319 PMID: 2924082
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Keywords: Arecaidine but-2-ynyl ester tosylate, Arecaidine but-2-ynyl ester tosylate supplier, Muscarinic, agonists, Receptors, Acetylcholine, Ach, butynyl, M2, 0382, Tocris Bioscience
Citations for Arecaidine but-2-ynyl ester tosylate
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