Arecaidine but-2-ynyl ester tosylate

Discontinued Product

Arecaidine but-2-ynyl ester tosylate (Cat. No. 0382) has been withdrawn from sale for commercial reasons.
Description: Muscarinic agonist
Chemical Name: N-Methyl-1,2,5,6-tetrahydropyridine-3-carboxylic acid but-2-ynyl ester tosylate
Literature (5)

Biological Activity for Arecaidine but-2-ynyl ester tosylate

Potent muscarinic agonist, 4.6-fold selective for M2 receptors in the atrium versus those in the ileum.

Technical Data for Arecaidine but-2-ynyl ester tosylate

M. Wt 365.44
Formula C11H15NO2.C7H8SO3
Storage Store at RT
CAS Number 119630-77-2
Smiles CC1=CC=C(C=C1)S(O)(=O)=O.CC#CCOC(=O)C1=CCCN(C)C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for Arecaidine but-2-ynyl ester tosylate

References for Arecaidine but-2-ynyl ester tosylate

References are publications that support the biological activity of the product.

Barlow and Weston-Smith (1985) The relative potencies of some agonists at M2 muscarinic receptors in guinea pig ileum, atria and bronchi. Br.J.Pharmacol. 85 437 PMID: 3896364

Moser et al (1989) Structure-activity relationships of new analogues of arecaidine propargyl ester at muscarinic M1 and M2 receptor subtypes. Br.J.Pharmacol. 96 319 PMID: 2924082

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Keywords: Arecaidine but-2-ynyl ester tosylate, Arecaidine but-2-ynyl ester tosylate supplier, Muscarinic, agonists, Receptors, Acetylcholine, Ach, butynyl, M2, 0382, Tocris Bioscience

Citations for Arecaidine but-2-ynyl ester tosylate

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Currently there are no citations for Arecaidine but-2-ynyl ester tosylate.

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