Arecaidine but-2-ynyl ester tosylate

Cat. No. 0382 Datasheet / COA / SDS

Discontinued Product

Unfortunately Arecaidine but-2-ynyl ester tosylate (Cat. No. 0382) has been withdrawn from sale for commercial reasons.
Cat.No. 0382 - Arecaidine but-2-ynyl ester tosylate | C11H15NO2.C7H8SO3 | CAS No. 119630-77-2
Description: Muscarinic agonist
Chemical Name: N-Methyl-1,2,5,6-tetrahydropyridine-3-carboxylic acid but-2-ynyl ester tosylate
Datasheet
Citations
Reviews
Literature

Biological Activity

Potent muscarinic agonist, 4.6-fold selective for M2 receptors in the atrium versus those in the ileum.

Technical Data

M. Wt 365.44
Formula C11H15NO2.C7H8SO3
Storage Store at RT
CAS Number 119630-77-2
Smiles CC1=CC=C(C=C1)S(O)(=O)=O.CC#CCOC(=O)C1=CCCN(C)C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Product Datasheets

Safety Datasheet

References

References are publications that support the products' biological activity.

Barlow and Weston-Smith (1985) The relative potencies of some agonists at M2 muscarinic receptors in guinea pig ileum, atria and bronchi. Br.J.Pharmacol. 85 437 PMID: 3896364

Moser et al (1989) Structure-activity relationships of new analogues of arecaidine propargyl ester at muscarinic M1 and M2 receptor subtypes. Br.J.Pharmacol. 96 319 PMID: 2924082

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Keywords: Arecaidine but-2-ynyl ester tosylate, supplier, Muscarinic, agonists, Receptors, Acetylcholine, Ach, butynyl, M2, Receptors, M2, Receptors, Tocris Bioscience

Citations for Arecaidine but-2-ynyl ester tosylate

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