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Submit Review5,7-Dichlorothiokynurenic acid
Discontinued Product
5,7-Dichlorothiokynurenic acid (Cat. No. 0296) has been withdrawn from sale for commercial reasons.
Description: Potent NMDA antagonist, acts glycine site
Chemical Name: 5,7-Dichloro-4-mercaptoquinoline-2-carboxylic acid
Biological Activity
NMDA receptor antagonist acting at the glycine site; reported to be more potent than the corresponding kynurenic acid analogue.
Technical Data
| M. Wt | 274.12 |
| Storage | Desiccate at -20°C |
| CAS Number | 135025-62-6 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets
Certificate of Analysis is currently unavailable on-line.
Please contact Customer Service
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References
References are publications that support the biological activity of the product.
Moroni et al (1991) Thiokynurenates: a new group of antagonists of the glycine modulatory site of the NMDA receptor. Eur.J.Pharmacol. 199 227 PMID: 1720099
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Keywords: 5,7-Dichlorothiokynurenic acid, 5,7-Dichlorothiokynurenic acid supplier, NMDA, Receptors, 0296, Tocris Bioscience
Citations for 5,7-Dichlorothiokynurenic acid
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