Cat. No. |
产品名称/活性 |
5867 |
Ceefourin 1 |
| Selective MRP4 inhibitor |
4193 |
CP 100356 hydrochloride |
| P-gp inhibitor |
4646 |
Elacridar hydrochloride |
| P-gp and BCRP inhibitor |
3241 |
Ko 143 |
| Potent and selective BCRP inhibitor |
4169 |
KS 176 |
| Selective BCRP inhibitor |
2338 |
MK 571 |
| MRP1 inhibitor; also CysLT1 (LTD4) inverse agonist |
2891 |
Ondansetron hydrochloride |
| Potent MATE1 inhibitor |
4107 |
Probenecid |
| MRP and OAT3 inhibitor |
4042 |
PSC 833 |
| Inhibitor of P-gp-mediated MDR |
3918 |
Pyrimethamine |
| Potent inhibitor of multidrug and toxin extrusion (MATE) transporters; also DHFR and STAT3 inhibitor |
3722 |
Reversan |
| Selective MRP1 and P-gp inhibitor |
5757 |
Tariquidar dihydrochloride |
| Potent P-glycoprotein (P-gp) inhibitor |
5456 |
Zosuquidar trihydrochloride |
| High affinity P-gp inhibitor |