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Submit ReviewVirodhamine trifluoroacetate
Description: TFA salt of virodhamine, an endogenous cannabinoid receptor mixed agonist/antagonist
Chemical Name: O-(2-Aminoethyl)-5Z,8Z,11Z,14Z-eicosatetraenoate trifluoroacetate
Purity: ≥98% (HPLC)
Biological Activity for Virodhamine trifluoroacetate
Virodhamine trifluoroacetate is a TFA salt of virodhamine, an endogenous cannabinoid receptor mixed agonist/antagonist that is found in higher concentrations peripherally than anandamide. Virodhamine is a full agonist at GPR55 and CB2 and partial agonist/antagonist at CB1 (EC50 values are 12, 381 and 2920 nM at GPR55, CB2 and CB1 receptors respectively).
Technical Data for Virodhamine trifluoroacetate
| M. Wt | 461.56 |
| Formula | C22H37NO2.CF3CO2H |
| Storage | Store at -20°C |
| Purity | ≥98% (HPLC) |
| CAS Number | 1415264-56-0 |
| PubChem ID | 91691131 |
| InChI Key | APQWCQIPZHJFAU-XVSDJDOKSA-N |
| Smiles | O=C(OCCN)CCC\C=C/C\C=C/C/C=C\C/C=C\CCCCC.FC(F)(F)C(O)=O |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for Virodhamine trifluoroacetate
References for Virodhamine trifluoroacetate
References are publications that support the biological activity of the product.
Porter et al (2002) Characterization of a novel endocannabinoid, virodhamine, with antagonist activity at the CB1 receptor. J.Pharmacol.Exp.Ther. 301 1020 PMID: 12023533
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1 Citation for Virodhamine trifluoroacetate
Citations are publications that use Tocris products. Selected citations for Virodhamine trifluoroacetate include:
Hayase (2013) Working memory- and anxiety-related behavioral effects of repeated nicotine as a stressor: the role of cannabinoid receptors. BMC Neurosci 14 20 PMID: 23394117
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Cannabinoid Receptor Ligands Scientific Review
Written by Roger Pertwee, this review discusses compounds which affect the activity of the endocannabinoid system, focusing particularly on ligands that are most widely used as experimental tools and denotes compounds available from Tocris.