PF9 tetrasodium salt

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Cat.No. 4074 - PF9 tetrasodium salt | C18H16N5Na4O13P3 | CAS No. 851265-78-6
Description: Potent GPR17 agonist
Chemical Name: 2-(Phenylethynyl)adenosine-5'-triphosphate tetrasodium salt
Purity: ≥98% (HPLC)
Datasheet
Citations
Literature

Biological Activity

Potent agonist of GPR17 (EC50 = 36 pM).

Technical Data

M. Wt 695.23
Formula C18H16N5Na4O13P3
Storage Store at -20°C
Purity ≥98% (HPLC)
CAS Number 851265-78-6
PubChem ID 90488909
InChI Key ONTPGXYSNYMMOK-YEJXUIBNSA-J
Smiles [Na+].[Na+].[Na+].[Na+].NC1=C2N=CN(C3O[C@H](COP([O-])(=O)OP([O-])(=O)OP([O-])([O-])=O)[C@@H](O)[C@H]3O)C2=NC(=N1)C#CC1=CC=CC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

SolubilitySoluble in water (supplied pre-dissolved at a concentration of 10mM)

Preparing Stock Solutions

The following data is based on the product molecular weight 695.23. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.44 mL 7.19 mL 14.38 mL
5 mM 0.29 mL 1.44 mL 2.88 mL
10 mM 0.14 mL 0.72 mL 1.44 mL
50 mM 0.03 mL 0.14 mL 0.29 mL

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Product Datasheets

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References

References are publications that support the products' biological activity.

Calleri et al (2010) Frontal affinity chromatography-mass spectrometry useful for characterization of new ligands for GPR17 receptor. J.Med.Chem. 53 3489 PMID: 20394377


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GPCR

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