Potent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). Exhibits >10,000-fold selectivity for hM3Dq over hM3.
|Storage||Store at RT|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
|Solvent||Max Conc. mg/mL||Max Conc. mM|
|water||1.46||5 with gentle warming|
Preparing Stock Solutions
The following data is based on the product molecular weight 291.39. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||3.43 mL||17.16 mL||34.32 mL|
|5 mM||0.69 mL||3.43 mL||6.86 mL|
|10 mM||0.34 mL||1.72 mL||3.43 mL|
|50 mM||0.07 mL||0.34 mL||0.69 mL|
References are publications that support the biological activity of the product.
Chen et al (2015) The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem.Neurosci. 6 476 PMID: 25587888
If you know of a relevant reference for Perlapine, please let us know.
Keywords: Perlapine, Perlapine supplier, Perlapine, potent, selective, hM3Dq, DREADD, agonists, antagonism, designer, receptors, drugs, muscarinic, activators, DREADDs, M3, Receptors, 5549, Tocris Bioscience
Citations for Perlapine
Citations are publications that use Tocris products.
Currently there are no citations for Perlapine. Do you know of a great paper that uses Perlapine from Tocris? Please let us know.
Reviews for Perlapine
There are currently no reviews for this product. Be the first to review Perlapine and earn rewards!
Have you used Perlapine?
Submit a review and receive an Amazon gift card.
$50/€35/£30/$50CAN/¥300 Yuan/¥5000 Yen for first to review with an image
$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image
Literature in this Area
Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* or download your copy today!
*Please note that Tocris will only send literature to established scientific business / institute addresses.