(±)-1-(1,2-Diphenylethyl)piperidine maleate

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Cat.No. 0360 - (±)-1-(1,2-Diphenylethyl)piperidine maleate | C19H23N.C4H4O4 | CAS No. 207461-99-2
Description: NMDA antagonist, acts ion channel site
Datasheet
Citations (1)
Reviews
Literature

Biological Activity

High affinity antagonist at the ion channel on the NMDA receptor.

Technical Data

M. Wt 381.47
Formula C19H23N.C4H4O4
Storage Store at RT
CAS Number 207461-99-2
PubChem ID 16657069
InChI Key AEHZEDLXDLPQQD-BTJKTKAUSA-N
Smiles OC(=O)\C=C/C(O)=O.C(C(N1CCCCC1)C1=CC=CC=C1)C1=CC=CC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

SolubilitySoluble to 10 mM in water

Preparing Stock Solutions

The following data is based on the product molecular weight 381.47. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.62 mL 13.11 mL 26.21 mL
5 mM 0.52 mL 2.62 mL 5.24 mL
10 mM 0.26 mL 1.31 mL 2.62 mL
50 mM 0.05 mL 0.26 mL 0.52 mL

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Product Datasheets

Safety Datasheet

References

References are publications that support the products' biological activity.

Ragawski (1993) Therapeutic potential of excitatory amino acid antagonists: channel blockers and 2,3-benzodiazepines. TiPS 14 325 PMID: 7504360


If you know of a relevant reference for (±)-1-(1,2-Diphenylethyl)piperidine maleate, please let us know.

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1 Citation for (±)-1-(1,2-Diphenylethyl)piperidine maleate

Citations are publications that use Tocris products. Selected citations for (±)-1-(1,2-Diphenylethyl)piperidine maleate include:

Ataka et al (2012) Alteration of antral and proximal colonic motility induced by chronic psychological stress involves central urocortin 3 and vasopressin in rats. Am J Physiol Gastrointest Liver Physiol 303 G519 PMID: 22651925


Do you know of a great paper that uses (±)-1-(1,2-Diphenylethyl)piperidine maleate from Tocris? If so please let us know.

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