Dihydroergocristine mesylate

Pricing Availability Delivery Time Qty
Cat.No. 0474 - Dihydroergocristine mesylate | C35H41N5O5.CH3SO3H | CAS No. 24730-10-7
Description: Partial α agonist. Non-selective
Chemical Name: (5'α,10α)-9,10-Dihydro-12'-hydroxy-2'-(1-methylethyl)-5'-(phenylmethyl)-ergotaman-3',6',18-trione mesylate
Purity: ≥98% (HPLC)
Datasheet
Citations
Literature

Biological Activity

5-HT receptor antagonist; partial agonist at adrenergic and dopaminergic receptors.

Compound Libraries

Dihydroergocristine mesylate is also offered as part of the Tocriscreen Plus. Find out more about compound libraries available from Tocris.

Technical Data

M. Wt 707.84
Formula C35H41N5O5.CH3SO3H
Storage Store at RT
Purity ≥98% (HPLC)
CAS Number 24730-10-7
PubChem ID 444034
InChI Key SPXACGZWWVIDGR-SPZWACKZSA-N
Smiles CS(=O)(O)=O.[H][C@]4([C@@]([H])3C[C@@H]([C@@](N[C@@]5([C@H](C)C)C(N([C@@]([H])(CC8=CC=CC=C8)C(N7[C@]([H])6CCC7)=O)[C@@]6(O)O5)=O)=O)CN4C)CC1=CNC2=C1C3=CC=C2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 17.7 25

Preparing Stock Solutions

The following data is based on the product molecular weight 707.84. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.41 mL 7.06 mL 14.13 mL
5 mM 0.28 mL 1.41 mL 2.83 mL
10 mM 0.14 mL 0.71 mL 1.41 mL
50 mM 0.03 mL 0.14 mL 0.28 mL

Molarity Calculator

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Reconstitution Calculator

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Product Datasheets

Safety Datasheet

References

References are publications that support the products' biological activity.

Drago (1988) Dihydroergocristine and memory alterations of aged male rats. Pharmacol.Biochem.Behav. 30 961 PMID: 3147464


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Citations for Dihydroergocristine mesylate

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Literature in this Area

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Pathways for Dihydroergocristine mesylate

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