BMY 45778

Discontinued Product

BMY 45778 (Cat. No. 1442) has been withdrawn from sale for commercial reasons.
Description: Non-prostanoid prostacyclin IP receptor partial agonist
Chemical Name: [3-(4,5-Diphenyl[2,4'-bioxazol]-5'-yl)phenoxy]acetic acid
Purity: ≥99% (HPLC)
Datasheet
Citations
Reviews
Literature (5)

Biological Activity for BMY 45778

BMY 45778 is a non-prostanoid prostacyclin mimetic that acts as a partial agonist at IP1 prostacyclin receptors. Potently inhibits platelet aggregation in vitro (IC50 = 27-35 nM).

Licensing Information

Sold with the permission of Bristol-Myers Squibb Company

Technical Data for BMY 45778

M. Wt 438.44
Formula C26H18N2O5
Storage Store at +4°C
Purity ≥99% (HPLC)
CAS Number 152575-66-1
PubChem ID 127861
InChI Key DSRSEEYZGWTODH-UHFFFAOYSA-N
Smiles OC(=O)COC1=CC(=CC=C1)C1=C(N=CO1)C1=NC(=C(O1)C1=CC=CC=C1)C1=CC=CC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for BMY 45778

Certificate of Analysis / Product Datasheet
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Keywords: BMY 45778, BMY 45778 supplier, Non-prostanoid, prostacyclin, IP1, receptor, partial, agonist, Receptors, Prostanoid, PGI, prostaglandins, prostacyclins, eicosanoids, BMY45778, 1442, Tocris Bioscience

Citations for BMY 45778

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Currently there are no citations for BMY 45778.

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Literature in this Area

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