Highly potent and selective androgen receptor (AR) agonist (EC50 = 0.44 nM). Exhibits selectivity for ARs over estrogen, glucocorticoid and mineralocorticoid receptors and no significant binding to steroid hormone binding globulin or aromatase. Also exhibits selectivity for muscle over prostate ARs. Active in vivo and orally bioavailable.
|Storage||Store at -20°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
|Solvent||Max Conc. mg/mL||Max Conc. mM|
Preparing Stock Solutions
The following data is based on the product molecular weight 305.72. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||3.27 mL||16.35 mL||32.71 mL|
|5 mM||0.65 mL||3.27 mL||6.54 mL|
|10 mM||0.33 mL||1.64 mL||3.27 mL|
|50 mM||0.07 mL||0.33 mL||0.65 mL|
References are publications that support the products' biological activity.
Ostrowski et al (2007) Pharmacological and X-ray structural characterization of a novel selective androgen receptor modulator: potent hyperanabolic stimulation of skeletal muscle with hypostimulation of prostate in rats. Endocrinology 148 4 PMID:
If you know of a relevant reference for BMS 564929, please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: BMS 564929, supplier, BMS564929, highly, potent, muscle-selective, androgen, receptor, AR, agonist, orally, bioavailable, Androgen, Receptor, Androgen, Receptor, Tocris Bioscience
Citations for BMS 564929
Citations are publications that use Tocris products.
Currently there are no citations for BMS 564929. Do you know of a great paper that uses BMS 564929 from Tocris? If so please let us know.
Reviews for BMS 564929
There are currently no reviews for this product. Be the first to review BMS 564929 and earn rewards!
Have you used BMS 564929?
Submit a review and receive an Amazon gift card.
$10US/$10CAN/€7/£6 gift card for a review without an image
$25US/$25CAN/€18/£15 gift card for a review with an image
*Offer only valid in the USA / Canada, UK and EuropeSubmit a Review
Literature in this Area
Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* or download your copy today!
*Please note that Tocris will only send literature to established scientific business / institute addresses.