5-Methoxy-N-cyclopropanoyltryptamine

Discontinued Product

Unfortunately 5-Methoxy-N-cyclopropanoyltryptamine (Cat. No. 0766) has been withdrawn from sale for commercial reasons.
Cat.No. 0766 - 5-Methoxy-N-cyclopropanoyltryptamine
Description: Melatonin agonist
Datasheet
Citations
Reviews
Literature

Biological Activity

A potent melatonin agonist which shows selectivity for melatonin binding sites in pars tuberalis (affinity 100-fold greater than melatonin) compared to avian brain (affinity 2-4 fold less than melatonin).

Licensing Information

Sold with the permission of ADIR et Cie.

Technical Data

M. Wt 258.32
Storage Desiccate at +4°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Preparing Stock Solutions

The following data is based on the product molecular weight 258.32. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.87 mL 19.36 mL 38.71 mL
5 mM 0.77 mL 3.87 mL 7.74 mL
10 mM 0.39 mL 1.94 mL 3.87 mL
50 mM 0.08 mL 0.39 mL 0.77 mL

Molarity Calculator

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Reconstitution Calculator

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Product Datasheets

Certificate of Analysis is currently unavailable
on-line. Please contact Customer Service
Safety Datasheet

References

References are publications that support the products' biological activity.

Depreux et al (1994) Synthesis and structure-activity relationships of novel naphthalenic and biosteric related amidic derivatives as melatonin receptor ligands. J.Med.Chem. 37 3231 PMID: 7932550

Spandoni et al (1993) 2-Substituted 5-methoxy-N-acyltryptamines: synthesis, binding affinity for the melatonin receptor and evaluation of the biological activity. J.Med.Chem. 36 4069 PMID: 8258829

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Keywords: 5-Methoxy-N-cyclopropanoyltryptamine, supplier, Melatonin, (MT), Receptors, Melatonin, (MT), Receptors, Tocris Bioscience

Citations for 5-Methoxy-N-cyclopropanoyltryptamine

Citations are publications that use Tocris products.

Currently there are no citations for 5-Methoxy-N-cyclopropanoyltryptamine.

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* or download your copy today!

*Please note that Tocris will only send literature to established scientific business / institute addresses.


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