4-[N-(4-Chlorophenyl)carbamoyloxy]-4-pent-2-ynyl-trimethyl ammonium iodide

Discontinued Product

Unfortunately 4-[N-(4-Chlorophenyl)carbamoyloxy]-4-pent-2-ynyl-trimethyl ammonium iodide (Cat. No. 0466) has been withdrawn from sale for commercial reasons.
Cat.No. 0466 - 4-[N-(4-Chlorophenyl)carbamoyloxy]-4-pent-2-ynyl-trimethylammonium iodide | CAS No. 141063-77-6
Description: Partial agonist at ganglionic M1 receptor
Datasheet
Citations
Reviews
Literature

Biological Activity

A partial agonist with 16 times the power of the analogue McN-A-343 in increasing arterial blood pressure and 18 times the affinity of the latter for ganglionic M1 receptors.

Technical Data

M. Wt 422.69
Storage Store at RT
CAS Number 141063-77-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Preparing Stock Solutions

The following data is based on the product molecular weight 422.69. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.37 mL 11.83 mL 23.66 mL
5 mM 0.47 mL 2.37 mL 4.73 mL
10 mM 0.24 mL 1.18 mL 2.37 mL
50 mM 0.05 mL 0.24 mL 0.47 mL

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Product Datasheets

Certificate of Analysis is currently unavailable
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Safety Datasheet

References

References are publications that support the products' biological activity.

Nilsson et al (1992) Amide, urea and carbamate analogues of the muscarinic agent [4-[[N-(3-chlorophenyl)carbamoyl]oxy]-2-butynyl]trimethylammonium chloride. J.Med.Chem. 35 2787 PMID: 1379640

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Keywords: 4-[N-(4-Chlorophenyl)carbamoyloxy]-4-pent-2-ynyl-trimethylammonium iodide, supplier, Non-selective, Muscarinics, Non-selective, Muscarinics, Tocris Bioscience

Citations for 4-[N-(4-Chlorophenyl)carbamoyloxy]-4-pent-2-ynyl-trimethyl ammonium iodide

Citations are publications that use Tocris products.

Currently there are no citations for 4-[N-(4-Chlorophenyl)carbamoyloxy]-4-pent-2-ynyl-trimethyl ammonium iodide.

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