Fentanyl citrate

Discontinued Product

3247 has been discontinued.

说明: Potent and selective μ agonist
别名: Phentanyl citrate
化学名: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate
纯度: ≥99% (HPLC)
说明书
引用文献
评论
文献 (2)

生物活性 for Fentanyl citrate

Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.

技术数据 for Fentanyl citrate

分子量 528.59
公式 C22H28N2O.C6H8O7
储存 Store at RT
纯度 ≥99% (HPLC)
CAS Number 990-73-8
PubChem ID 13810
InChI Key IVLVTNPOHDFFCJ-UHFFFAOYSA-N
Smiles O=C(O)C(O)(CC(O)=O)CC(O)=O.O=C(CC)N(C3=CC=CC=C3)C1CCN(CCC2=CC=CC=C2)CC1

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for Fentanyl citrate

参考文献 for Fentanyl citrate

参考文献是支持产品生物活性的出版物。

Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113 PMID: 7475964

Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233 PMID: 12738037

Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054 PMID: 14557380

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关键词: Fentanyl citrate, Fentanyl citrate supplier, Potent, selective, μ-opioid, mu-opioid, agonists, MOP, Receptors, OP3, Phentanyl, citrate, Mu, Opioid, 3247, Tocris Bioscience

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