JAK Inhibitors
| Cat. No. | 产品名称/活性 |
|---|---|
| 0414 | AG 490 |
| JAK2, JAK3 inhibitor. Also EGFR-kinase inhibitor | |
| 7222 | Baricitinib |
| Highly potent JAK1 and JAK2 inhibitor; also inhibits JAK3 and Tyk2 | |
| 4556 | CP 690550 citrate |
| Potent JAK inhibitor | |
| 3395 | Lestaurtinib |
| JAK2, FLT3 and TrkA inhibitor; also inhibits AurA and AurB | |
| 6506 | PF 06551600 malonate |
| Potent and selective JAK3 inhibitor | |
| 6577 | Pyridone 6 |
| Potent pan-JAK inhibitor; induces intermediate mesoderm; cell-permeable | |
| 7064 | Ruxolitinib |
| Potent and selective JAK1/JAK2 inhibitor; orally bioavailable | |
| 7048 | Ruxolitinib phosphate |
| Phosphate salt of Ruxolitinib (Cat. No. 7064); potent and selective JAK1/JAK2 inhibitor | |
| 3035 | SD 1008 |
| JAK2/STAT3 signaling pathway inhibitor | |
| 6125 | TC JL 37 |
| Potent TYK2 inhibitor | |
| 7783 | Upadacitinib |
| JAK1-selective inhibitor |