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Submit ReviewRVD-Hpα
说明： Selective CB1 agonist; also CB2 PAM
别名： Pepcan-12
生物活性 for RVD-Hpα
RVD-Hpα is a N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM).
技术数据 for RVD-Hpα
| 分子量 | 1424.66 |
| 公式 | C65H105N19O17 |
| 序列 | RVDPVNFKLLSH |
| 储存 | Store at -20°C |
| CAS Number | 1193362-76-3 |
| PubChem ID | 90488874 |
| InChI Key | CSDQEWILNKOWRN-WSDCEOHFSA-N |
| Smiles | [H]N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC1=CNC=N1)C(O)=O |
上方提供的技术数据仅供参考。批次相关数据请参见分析证书。
Tocris products are intended for laboratory research use only, unless stated otherwise.
产品说明书 for RVD-Hpα
参考文献 for RVD-Hpα
参考文献是支持产品生物活性的出版物。
Gomes et al (2009) Novel endogenous peptide agonists of cannabinoid receptors. FASEB J. 23 3020 PMID: 19380512
Khurana et al (2017) Modulation of CB1 cannabinoid receptor by allosteric ligands: Pharmacology and therapeutic opportunities. Neuropharmacology 124 3 PMID: 28527758
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关键词: RVD-Hpalpha, RVD-Hpalpha supplier, selective, CB1, receptors, agonists, cannabinoids, RVD-Hpalpha, RVD-Hpα, cb1r, high, affinity, CB2, positive, allosteric, modulator, PAM, endocannabinoids, Pepcan-12, Receptors, 3744, Tocris Bioscience
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*请注意，Tocris 仅会向正规科研企业/机构地址发送文献。
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