WAY 207024 dihydrochloride

Name: WAY 207024 dihydrochloride
Brand: Tocris Bioscience
SKU: 3890

Cat. No. 3890 提交评论说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

3890 has been discontinued.

View all Gonadotropin-Releasing Hormone Receptors products.

说明： GnRH receptor antagonist

化学名： 6-[[4-[2-[4-(1,1-Dimethylethyl)phenyl]-1H-benzimidazol-7-yl]-i-piperazinyl]methyl]-quinoxaline dihydrochloride

纯度： ≥99% (HPLC)

说明书

引用文献

生物活性技术数据说明书参考文献

生物活性 for WAY 207024 dihydrochloride

WAY 207024 dihydrochloride is a gonadotropin releasing hormone receptor (GnRH-R) antagonist. Exhibits potent affinity (IC₅₀ values are 12 and 71 nM for human and rat GnRH receptors respectively). Lowers plasma leuteinizing hormone levels in the rat. Orally active.

许可信息

Sold for research purposes under agreement from Pfizer Inc.

技术数据 for WAY 207024 dihydrochloride

分子量	549.54
公式	C₃₀H₃₂N₆.2HCl
储存	Desiccate at RT
纯度	≥99% (HPLC)
CAS Number	872002-73-8
PubChem ID	69403574
InChI Key	REQCNTGYEABOIT-UHFFFAOYSA-N
Smiles	CC(C)(C)C(C=C6)=CC=C6C(N5)=NC1=C5C(N(CC4)CCN4CC2=CC=C(N=CC=N3)C3=C2)=CC=C1.Cl.Cl

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

产品说明书 for WAY 207024 dihydrochloride

分析证书/产品说明书

化学品安全技术说明书

参考文献 for WAY 207024 dihydrochloride

参考文献是支持产品生物活性的出版物。

Pelletier et al (2009) Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the g.tropin releasing hormone receptor (GnRH-R). J.Med.Chem. 52 214 PMID: 19072222

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篇 WAY 207024 dihydrochloride 的引用文献

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