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Virodhamine

Cat. No. 1569 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

1569 has been discontinued.

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说明： GPR55 and CB2 agonist. CB1 partial agonist/antagonist
别名： O-Arachidonyl ethanolamine
化学名： O-(2-Aminoethyl)-5Z,8Z,11Z,14Z-eicosatetraenoate
说明书
引用文献
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生物活性 技术数据 说明书 参考文献

生物活性 for Virodhamine

Endogenous cannabinoid receptor mixed agonist/antagonist found in higher concentrations peripherally than anandamide. Full agonist at GPR55 and CB2 and partial agonist/antagonist at CB1 (EC50 values are 12, 381 and 2920 nM at GPR55, CB2 and CB1 receptors respectively). Induces hypothermia in vivo.

技术数据 for Virodhamine

分子量 347.54
公式 C22H37NO2
储存 Desiccate at -20°C
CAS Number 287937-12-6
Smiles O=C(OCCN)CCC\C=C/C\C=C/C/C=C\C/C=C\CCCCC

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

参考文献 for Virodhamine

参考文献是支持产品生物活性的出版物。

Porter et al (2002) Characterization of a novel endocannabinoid, virodhamine, with antagonist activity at the CB1 receptor. J.Pharmacol.Exp.Ther. 301 1020 PMID: 12023533

Ryberg et al (2007) The orphan receptor GPR55 is a novel cannabinoid receptor. Br.J.Pharmacol. 152 1092 PMID: 17876302

Sauer et al (2002) Further characterization of the novel endocannabinoid virodhamine. 2002 Symposium on the Cannabinoids, International

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关键词: Virodhamine, Virodhamine supplier, GPR55, CB2, agonists, CB1, partial, antagonists, non-selective, cannabinoids, receptors, cb2r, cb1r, O-Arachidonyl, ethanolamine, Non-selective, Cannabinoids, 1569, Tocris Bioscience

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该领域的文献

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Cannabinoid Receptor Ligands Scientific Review

Cannabinoid Receptor Ligands Scientific Review

Written by Roger Pertwee, this review discusses compounds which affect the activity of the endocannabinoid system, focusing particularly on ligands that are most widely used as experimental tools and denotes compounds available from Tocris.