Talsupram hydrochloride

Cat. No. 4352 提交评论说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

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大包装订单

Cat.No. 4352 - Talsupram hydrochloride | C20H25NS.HCl | CAS No. 25487-28-9

说明： Selective inhibitor of noradrenalin transporters

化学名： 1,3-Dihydro-N,3,3-trimethyl-1-phenylbenzo[c]thiophene-1-propanamine hydrochloride

纯度： ≥98% (HPLC)

文献 (1)

生物活性技术数据溶解性计算器说明书参考文献

生物活性 for Talsupram hydrochloride

Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor; exhibits a high affinity for the human noradrenalin transporter (NET) against SERT and DAT (IC₅₀ values are 0.79, 850 and 9300 nM for inhibition of monoamine uptake by NET, SERT and DAT respectively). Antidepressant.

技术数据 for Talsupram hydrochloride

分子量	347.95
公式	C₂₀H₂₅NS.HCl
储存	Desiccate at RT
纯度	≥98% (HPLC)
CAS Number	25487-28-9
PubChem ID	33013
InChI Key	YMZCMCDSCRSIBS-UHFFFAOYSA-N
Smiles	CC2(C)SC(C3=CC=CC=C3)(CCCNC)C1=CC=CC=C12.Cl

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

溶解性数据 for Talsupram hydrochloride

	溶剂	最高浓度 mg/mL	最高浓度 mM
溶解性
	water	6.96	20
	DMSO	34.8	100

制备储备液 for Talsupram hydrochloride

以下数据基于产品分子量 347.95。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

浓度/溶剂体积/质量	1 mg	5 mg	10 mg
1 mM	2.87 mL	14.37 mL	28.74 mL
5 mM	0.57 mL	2.87 mL	5.75 mL
10 mM	0.29 mL	1.44 mL	2.87 mL
50 mM	0.06 mL	0.29 mL	0.57 mL

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产品说明书 for Talsupram hydrochloride

分析证书/产品说明书

化学品安全技术说明书

参考文献 for Talsupram hydrochloride

参考文献是支持产品生物活性的出版物。

McConathy et al (2004) Synthesis and biological evaluation of [¹¹C]talopram and [¹¹C]talsupram: candidate PET ligands for the NE transporter. Nucl.Med.Biol. 31 705 PMID: 15246361

Schou et al (2006) Synthesis and positron emission tomography evaluation of three NE transporter radioligands: [C-11]desipramine, [C-11]talopram and [C-11]talsupram. Mol.Imaging Biol. 8 1

Rowlett et al (2004) Cocaine-like discriminative stimulus effects of heroin: modulation by selective monoamine transport inhibitors. J.Pharmacol.Exp.Ther. 310 342 PMID: 14985417

If you know of a relevant reference for Talsupram hydrochloride, please let us know.

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