Talsupram hydrochloride

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Cat.No. 4352 - Talsupram hydrochloride | C20H25NS.HCl | CAS No. 25487-28-9
说明: Selective inhibitor of noradrenalin transporters
化学名: 1,3-Dihydro-N,3,3-trimethyl-1-phenylbenzo[c]thiophene-1-propanamine hydrochloride
纯度: ≥98% (HPLC)
文献 (1)

生物活性 for Talsupram hydrochloride

Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor; exhibits a high affinity for the human noradrenalin transporter (NET) against SERT and DAT (IC50 values are 0.79, 850 and 9300 nM for inhibition of monoamine uptake by NET, SERT and DAT respectively). Antidepressant.

技术数据 for Talsupram hydrochloride

分子量 347.95
公式 C20H25NS.HCl
储存 Desiccate at RT
纯度 ≥98% (HPLC)
CAS Number 25487-28-9
PubChem ID 33013
Smiles CC2(C)SC(C3=CC=CC=C3)(CCCNC)C1=CC=CC=C12.Cl


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溶解性数据 for Talsupram hydrochloride

溶剂 最高浓度 mg/mL 最高浓度 mM
water 6.96 20
DMSO 34.8 100

制备储备液 for Talsupram hydrochloride

以下数据基于产品分子量 347.95。 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

浓度/溶剂体积/质量 1 mg 5 mg 10 mg
1 mM 2.87 mL 14.37 mL 28.74 mL
5 mM 0.57 mL 2.87 mL 5.75 mL
10 mM 0.29 mL 1.44 mL 2.87 mL
50 mM 0.06 mL 0.29 mL 0.57 mL

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产品说明书 for Talsupram hydrochloride

参考文献 for Talsupram hydrochloride


McConathy et al (2004) Synthesis and biological evaluation of [11C]talopram and [11C]talsupram: candidate PET ligands for the NE transporter. Nucl.Med.Biol. 31 705 PMID: 15246361

Schou et al (2006) Synthesis and positron emission tomography evaluation of three NE transporter radioligands: [C-11]desipramine, [C-11]talopram and [C-11]talsupram. Mol.Imaging Biol. 8 1

Rowlett et al (2004) Cocaine-like discriminative stimulus effects of heroin: modulation by selective monoamine transport inhibitors. J.Pharmacol.Exp.Ther. 310 342 PMID: 14985417

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