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KuWal151

Cat. No. 6644 提交评论 说明书 / 分析证书（CoA） / 化学品安全技术说明书（SDS）

Discontinued Product

6644 has been discontinued.

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说明： Potent and selective CLK inhibitor
化学名： 3-(3-Chlorophenyl)-6,7-dihydropyrrolo[3,4-g]indol-8(1H)-one
纯度： ≥98% (HPLC)
说明书
引用文献
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生物活性 技术数据 说明书 参考文献

生物活性 for KuWal151

KuWal151 is a potent and selective CLK inhibitor (IC50 values are 28, 88 and 510 nM for CLK4, 1 and 2, respectively). Exhibits no significant activity at CLK3, DYRK, CDK or GSK3 at a concentration of 10 μM. Inhibits growth of a range of cancer cell lines in vitro at subnanomolar concentrations.

技术数据 for KuWal151

分子量 282.72
公式 C16H11ClN2O
储存 Store at +4°C
纯度 ≥98% (HPLC)
CAS Number 2341841-06-1
Smiles O=C1C2=C(CN1)C=CC3=C2NC=C3C4=CC=CC(Cl)=C4

上方提供的技术数据仅供参考。批次相关数据请参见分析证书。

Tocris products are intended for laboratory research use only, unless stated otherwise.

参考文献 for KuWal151

参考文献是支持产品生物活性的出版物。

Walter et al (2018) Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype. PLoS One 13 e0196761 PMID: 29723265

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关键词: KuWal151, KuWal151 supplier, Clk, inibitors, inhibits, Cdc2-like, kinases, selective, potent, anticancer, CLK, (Cdc2-like, kinases), 6644, Tocris Bioscience

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