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Home » Pharmacology » All Targets
All Targets
Pharmacological targets listed alphabetically
κBA1 ReceptorsA2A ReceptorsA2B ReceptorsA3 ReceptorsAbl KinaseACATACEAcetylcholine Muscarinic ReceptorsAcetylcholine Nicotinic ReceptorsAcetylcholine, OtherAcetylcholine α4β2 Nicotinic ReceptorsAcetylcholine α7 Nicotinic ReceptorsAcetylcholine Nicotinic Receptors, Non-SelectiveAcetylcholine Nicotinic Receptors, Other SubtypesAcetylcholinesteraseAcetylcholine TransportersAChEAcid sensing ion channel 3ActinActivator Protein-1Activin Receptor-like KinaseAcyl-CoA:cholesterol acyltransferaseAcyltransferasesAdenine ReceptorsAdenine ReceptorsAdenosine, OtherAdenosine A1 ReceptorsAdenosine A2A ReceptorsAdenosine A2B ReceptorsAdenosine A3 ReceptorsAdenosine DeaminaseAdenosine KinaseAdenosine ReceptorsAdenosine TransportersAdenosine UptakeAdenylyl CyclaseADKAdrenergic α1 ReceptorsAdrenergic α2 ReceptorsAdrenergic Alpha Receptors, Non-SelectiveAdrenergic β1 ReceptorsAdrenergic β2 ReceptorsAdrenergic β3 ReceptorsAdrenergic Beta Receptors, Non-SelectiveAdrenergic ReceptorsAdrenergic Related CompoundsAdrenergic TransportersAdrenoceptorsAHRAkt (Protein Kinase B)Alcohol DehydrogenaseAldehyde DehydrogenaseAldehyde ReductaseAldose ReductaseAldosterone ReceptorsALK Receptors
Alpha-GlucosidaseAlpha-MannosidaseAlpha4Beta2 Nicotinic ReceptorsAlpha7 Nicotinic ReceptorsAlpha1 Adrenergic ReceptorsAlpha2 Adrenergic ReceptorsAminopeptidaseAMP-Activated Protein KinaseAMPA ReceptorsAMPKAMTAmylin ReceptorsAmyloid β Peptides Amyloid Precursor ProteinAMY ReceptorsAnandamide AmidaseAnandamide TransportersAndrogen ReceptorsAngiogenesisAngiotensin-Converting EnzymeAngiotensin AT1 ReceptorsAngiotensin AT2 ReceptorsAngiotensin ReceptorsAngiotensin Receptors, Non-SelectiveAnkyrin ReceptorsAnnexinANP ReceptorsAntiangiogenicsAntibioticsAntibodiesAntioxidantsAntiprionAntiviralsAP-1Apelin ReceptorsAPJ ReceptorsApoptosisApoptosis, OtherApoptosis InducersAPP SecretaseAromatic L-Amino Acid DecarboxylaseAryl Hydrocarbon ReceptorsASIC3AT1 ReceptorsAT2 ReceptorsAtaxia Telangiectasia and Rad3 Related KinaseAtaxia Telangiectasia Mutated KinaseATM and ATR KinasesATPaseATPases/GTPasesAT Receptors, Non-SelectiveAtrial Natriuretic Peptide ReceptorsATR KinaseAurora KinaseAutophagyAutotaxinAXOR12 Receptors
c-Ablc-Fosc-IAPc-RafC3Ca2+-Activated Potassium (KCa) ChannelsCa2+-ATPaseCaV ChannelsCa2+ Binding Protein ModulatorsCa2+ ChannelsCa2+ IonophoreCa2+Sensitive Protease ModulatorsCa2+ SignalingCa2+ Signaling Agents, GeneralCaged CompoundsCalcineurinCalcitonin and Related ReceptorsCalcium (CaV) ChannelsCalcium-ATPaseCalcium-Sensing ReceptorCalcium-Sensitive Protease ModulatorsCalcium Binding Protein ModulatorsCalcium ChannelsCalcium Channels, OtherCalcium IonophoreCalcium SignalingCalcium Signaling Agents, GeneralCalmodulinCalmodulin-Activated Protein KinaseCalpainCaM KinaseCaM Kinase KinasecAMPCannabinoid (CB1) ReceptorsCannabinoid (CB2) ReceptorsCannabinoid (GPR55) ReceptorsCannabinoid, Non-SelectiveCannabinoid, OtherCannabinoid ReceptorsCannabinoid TransportersCarbohydrate MetabolismCarboxypeptidaseCarrier ProteinCasein Kinase 1Casein Kinase 2CaspaseCASRCatechol-O-methyltransferaseCathepsinCB1 ReceptorsCB2 ReceptorsCCK-Inactivating Serine ProteaseCCK1 ReceptorsCCK2 ReceptorsCCK ReceptorsCCRcdc7Cdc25 PhosphataseCdk
Cell Adhesion MoleculesCell CycleCell Cycle InhibitorsCell MetabolismCell SignalingCellular ProcessesCeramidaseCeramide-Specific GlycosyltransferaseCFTRCGRP ReceptorsChannel Modulators, OtherCheckpoint Control KinasesCheckpoint KinaseChemokine ReceptorsChk1Chk2Chloride ChannelsCholecystokinin ReceptorsCholecystokinin, Non-SelectiveCholecystokinin1 ReceptorsCholecystokinin2 ReceptorsCholinesterasesChymaseCK1CK2Cl- ChannelscMETComplementCOMTConnexinsConvertase, C3-Corticotropin-Releasing Factor, Non-SelectiveCorticotropin-Releasing Factor1 ReceptorsCorticotropin-Releasing Factor2 ReceptorsCorticotropin-Releasing Factor ReceptorsCOXCRF, Non-SelectiveCRF1 ReceptorsCRF2 ReceptorsCRF ReceptorsCRTH2CT ReceptorsCXCRCyclasesCyclic Adenosine MonophosphateCyclic Nucleotide Dependent-Protein KinaseCyclin-Dependent Protein KinaseCyclooxygenaseCYPCysLT1 ReceptorsCysLT2 ReceptorsCysteinyl Aspartate ProteaseCytidine DeaminaseCytochrome P450Cytokine and NF-κB SignalingCytokine ReceptorsCytokinesCytoskeleton & Motor Proteins
D1 and D5 ReceptorsD2 ReceptorsD3 ReceptorsD4 ReceptorsDAG KinaseDAGLDATDeacetylasesDeaminasesDeath Domain Receptor-Associated Adaptor KinaseDecarboxylasesDehydrogenasesΔ7-Dehydrocholesterol ReductaseDelta Opioid ReceptorsDeoxycytidine KinaseDGAT-1DGKDHCRDHFRDiacylglycerolacyltransferase 1Diacylglycerol KinaseDiacylglycerol LipaseDihydrofolate Reductase
Dihydrotestosterone ReceptorsDipeptidaseDipeptidyl Peptidase IVDNA, RNA and Protein SynthesisDNA-Dependent Protein KinaseDNA-PKDNA LigaseDNA methyltransferaseDNA TopoisomeraseDopamine D1 ReceptorsDopamine D2-like, Non-SelectiveDopamine D2 ReceptorsDopamine D3 ReceptorsDopamine D4 ReceptorsDopamine D5 ReceptorsDopamine ReceptorsDopaminergic-RelatedDopamine TransportersDOP ReceptorsDPP-IVDP ReceptorsDual-Specificity PhosphataseDynamin
E-Type ATPaseEAATECEEcto-ATPaseEDG ReceptorsEGFRElastaseElk3ENaCEncephalitogenic Myelin Oligodendrocyte GlycoproteinEncephalitogenic Myelin Proteolipid FragmentEndocytosisEndopeptidase 24.15Endothelial LipaseEndothelial Nitric Oxide SynthaseEndothelin, Non-SelectiveEndothelin-Converting EnzymeETA ReceptorsETB ReceptorsEndothelin ReceptorseNOSENPP2ENT1Enzyme-Associated ReceptorsEnzyme-Linked Receptors
EnzymesEnzyme Substrates / ActivatorsEP1-4 ReceptorsEpacEpidermal Growth Factor ReceptorsEpithelial Sodium ChannelsEquilibrative Nucleoside TransportersERErbBERKERRE SelectinEsterasesEstrogen (GPR30) ReceptorsEstrogen ReceptorsET, Non-SelectiveETA ReceptorsETB ReceptorsET ReceptorsExcitatory Amino Acid TransportersExocytosisExonucleasesExtracellular Matrix and Adhesion MoleculesExtracellular Signal-Regulated Kinase
G-Protein-Coupled ReceptorsGβγGi/oGq/11GsGABA, MiscellaneousGABA-TransferaseGABAA and GABAC ReceptorsGABAA ReceptorsGABAB ReceptorsGABAC ReceptorsGABA TransportersGalanin ReceptorsGAL ReceptorsGamma-SecretaseGap ChannelsGastric Inhibitory Peptide ReceptorsGastrin-Releasing Peptide-Preferring ReceptorsGATGCPGeneral Calcium Signaling AgentsGeneral ImidazolinesGeranylgeranyltransferaseGhrelin ReceptorsGHS-R1a ReceptorsGIP ReceptorsGLASTGLP1 ReceptorsGLP2 ReceptorsGLT-1Glucagon-Like Peptide 1 ReceptorsGlucagon-Like Peptide 2 ReceptorsGlucagon and Related ReceptorsGlucagon ReceptorsGlucocorticoid ReceptorsGlucose-Dependent Insulinotropic PeptideGlucosidaseGlutamate (AMPA) Receptors
Glutamate (Ionotropic), Non-SelectiveGlutamate (Ionotropic) ReceptorsGlutamate (Kainate) ReceptorsGlutamate (Metabotropic) Group III ReceptorsGlutamate (Metabotropic) Group II ReceptorsGlutamate (Metabotropic) Group I ReceptorsGlutamate (Metabotropic) ReceptorsGlutamate (NMDA) ReceptorsGlutamate, MiscellaneousGlutamate Carboxypeptidase IIGlutamate (EAAT) TransportersGlutathione S-TransferaseGlycine ReceptorsGlycine TransportersGlycogen PhosphorylaseGlycogen Synthase Kinase 3Glycoprotein IIb/IIIa (αIIbα3)GlycosylasesGlycosyltransferaseGlyRGlyTGnRH ReceptorsGonadotrophin-Releasing Hormone ReceptorsGPCRGPR30 ReceptorsGPR40 ReceptorsGPR54 ReceptorsGPR55 ReceptorsGPR109 ReceptorsGPR119 ReceptorsG Proteins (Heterotrimeric)G Proteins (Small)Growth Factor ReceptorsGrowth Hormone Secretagog Receptor 1aGRP-Preferring ReceptorsGSKGTPaseGuanylyl Cyclase
H+, K+-ATPaseH+-ATPaseH1 ReceptorsH2 ReceptorsH3 ReceptorsH4 ReceptorsHDACHeat Shock Protein 70Heat Shock Protein 90Heat Shock ProteinsHedgehog SignalingHeme OxygenaseHeparanaseHepatocyte Growth Factor ReceptorsHerhERG ChannelsHexokinaseHexosaminidase, BetaHGFRHh SignalingHistamine H1 ReceptorsHistamine H2 ReceptorsHistamine H3 ReceptorsHistamine H4 Receptors
Histamine N-methyltransferaseHistamine ReceptorsHistaminergic-Related CompoundsHistone DeacetylaseHM74 ReceptorsHMG-CoA ReductaseHormone-sensitive LipasehOT7T175 ReceptorsHSLHsp70Hsp90HspsHuman Ether-A-Go-Go Related Gene ChannelsHuman Leukocyte ElastaseHuman Neutrophil ElastaseHydrogen, Potassium-ATPaseHydrogen-ATPaseHydrolasesHydroxylase, 11-βHydroxylasesHydroxysteroid Dehydrogenase, 11β-Hydroxytryptamine, 5- ReceptorsHydroxytryptamine, 5- Transporters
I1 ReceptorsI2 ReceptorsI3 ReceptorsIAPICAMIGF ReceptorsiGlu ReceptorsIκB KinaseIKKIL ReceptorsImidazoline (I1) ReceptorsImidazoline (I2) ReceptorsImidazoline (I3) ReceptorsImidazoline, GeneralImidazoline ReceptorsImmunosuppressantsIMPaseInducible Nitric Oxide SynthaseInhibitor of ApoptosisInhibitor of Kappa BiNOS
Inositol 1,4,5-triphosphate ReceptorsInositol and cAMP SignalingInositol LipidsInositol MonophosphataseInositol PhosphataseIns(1,4,5)P3 5-PhosphataseInsulin and Insulin-like ReceptorsIntegrin ReceptorsInterleukin ReceptorsInterleukinsInward Rectifier Potassium (KIR) ChannelsIon ChannelsIonophoresIonotropic Glutamate ReceptorsIon Pumps, OtherIon Pumps/TransportersIon TransportersIon Transporters, OtherIP3 ReceptorsIP ReceptorsIsomerases
M1 ReceptorsM2 ReceptorsM3 ReceptorsM4 ReceptorsM5 ReceptorsMAGLMammalian Target of RapamycinMannosidaseMAOMAPKMAPK, OtherMAPK SignalingMatrixinsMatrix MetalloproteaseMatrix Metalloproteinase (MMP)Maxi-K ChannelsMBOATMCH ReceptorsMcl-1MC ReceptorsMDM2MDRMEKMelanin-Concentrating Hormone ReceptorsMelanocortin (MC) ReceptorsMelastatin ReceptorsMelatonin ReceptorsMembrane-bound O-acyltransferase (MBOAT)Membrane Transport ProteinMET ReceptorsMetabotropic Glutamate ReceptorsMetastin ReceptorsMethionine Aminopeptidase-2MethyltransferasesmGlu, Non-SelectivemGlu1 ReceptorsmGlu2 ReceptorsmGlu3 ReceptorsmGlu4 ReceptorsmGlu5 ReceptorsmGlu6 ReceptorsmGlu7 Receptors
mGlu8 ReceptorsmGlu Group III ReceptorsmGlu Group II ReceptorsmGlu Group I ReceptorsmGlu ReceptorsMicrotubulesMineralocorticoid ReceptorsMiscellaneous OpioidsMiscellaneous CompoundsMiscellaneous GABAMiscellaneous GlutamateMitochondrial HexokinaseMitogen-Activated Protein KinaseMitogen-Activated Protein Kinase-Activated Protein Kinase-2Mitogen-Activated Protein Kinase KinaseMitosisMitotic Kinesin Eg5MK-2MLCKMMPMnk1Monoacylglycerol LipaseMonoamine OxidaseMonoamine TransportersMOP ReceptorsMotilin ReceptorsMotor ProteinsMre11-Rad50-Nbs1MRN ExonucleasemTORMT ReceptorsMultidrug TransportersMu Opioid ReceptorsMuscarinic (M1) ReceptorsMuscarinic (M2) ReceptorsMuscarinic (M3) ReceptorsMuscarinic (M4) ReceptorsMuscarinic (M5) ReceptorsMuscarinic ReceptorsMYCMyosinMyosin Light Chain Kinase
N-Methyl-D-Aspartate ReceptorsN-Myristoyltransferase-1N-Type Calcium ChannelsNa+/Ca2+ ExchangerNaV ChannelsNa+/2Cl-/K+ CotransporterNa+ ChannelsNAAG PeptidaseNAALADasenAChRNatriuretic Peptide ReceptorsNCAMNeovascularizationNETNetNeurokinin ReceptorsNeurolysinNeuromedin B-Preferring ReceptorsNeuromedin U ReceptorsNeuronal MetabolismNeuronal Nitric Oxide SynthaseNeuropeptide FF/AF ReceptorsNeuropeptide Y ReceptorsNeurotensin ReceptorsNeurotransmitter TransportersNeurotrophin ReceptorsNeutrophil ElastaseNF-κB & IκBNHE-1Nicotinic (α4β2) ReceptorsNicotinic (α7) ReceptorsNicotinic Acid ReceptorsNicotinic ReceptorsNicotinic Receptors (Non-Selective)Nicotinic Receptors (Other Subtypes)Nitric Oxide, OtherNitric Oxide detection reagentsNitric Oxide DonorsNitric Oxide PrecursorsNitric Oxide SignalingNitric Oxide SynthaseNitric Oxide Synthase, Non-SelectiveNK1 ReceptorsNK2 ReceptorsNK3 ReceptorsNKCC Cotransporter
NMB-Preferring ReceptorsNMDA ReceptorsNME2NMU ReceptorsnNOSNociceptin ReceptorsNO detectionNO Detection ReagentsNO Donors / PrecursorsNogo-66 ReceptorsNon-Selective / Other Potassium ChannelsNon-selective 5-HTNon-selective 5-HT1Non-selective 5-HT2Non-selective AdenosineNon-selective Adrenergic α ReceptorsNon-selective Adrenergic β ReceptorsNon-selective AT ReceptorsNon-selective CannabinoidsNon-selective CCKNon-selective CRFNon-selective DopamineNon-selective EndothelinNon-Selective Ionotropic GlutamateNon-selective Metabotropic GlutamateNon-Selective MuscarinicsNon-selective NOSNon-selective OrexinNon-selective PPARNOP ReceptorsNO PrecursorsNoradrenalin TransporterNO Synthase, Non-SelectiveNO SynthasesNotch SignalingNPFF ReceptorsNPP2NPRNPY ReceptorsNTPDaseNT ReceptorsNuclear Factor Kappa BNuclear ReceptorsNuclear Receptors, OtherNucleoside Transporters
O-GlcNAcaseOATP1B1OP1 ReceptorsOP2 ReceptorsOP3 ReceptorsOP4 ReceptorsOpioid, δ-Opioid, κ-Opioid, μ-Opioid ReceptorsOrexin, Non-SelectiveOrexin1 ReceptorsOrexin2 ReceptorsOrexin ReceptorsOrganic Anion Transporting PolypeptideORL1 ReceptorsOrnithine DecarboxylaseOrphan 7-TM ReceptorsOrphan 7-Transmembrane ReceptorsOrphan G-Protein-Coupled ReceptorsOrphan GPCRsOther AcetylcholineOther AdenosineOther ApoptosisOther ATPasesOther Calcium ChannelsOther CannabinoidsOther Channel ModulatorsOther Dehydrogenases
Other HydrolasesOther Ion Pumps/TransportersOther KinasesOther MAPKOther Nitric OxideOther Nuclear ReceptorsOther Oxygenases/OxidasesOther Peptide ReceptorsOther PharmacologyOther Product TypesOther ProteasesOther ReductasesOther RTKsOther Synthases/SynthetasesOther TachykininOther Transcription FactorsOther TransferasesOther TRP ChannelsOther Wnt SignalingOT ReceptorsOX1 ReceptorsOX2 ReceptorsOXE ReceptorsOxidaseOxidative PhosphorylationOxoeicosanoid receptorsOxygenases/OxidasesOxytocin Receptors
P-GlycoproteinP-SelectinP-Type ATPaseP-Type Calcium ChannelsP2X ReceptorsP2Y Receptorsp14ARFp38 MAPKp53p56lckp60c-srcp70 S6Kp75p90 Ribosomal S6 Kinasep160ROCKPAC1 ReceptorsPACAP ReceptorsPAF ReceptorsPAOParathyroid Hormone ReceptorsPARPPAR ReceptorsPC-PLCPDEPDGFRPDK1PDPK1Peptide Receptor, OtherPeptide ReceptorsPeroxisome-Proliferating ReceptorsPGFPGI2Phenylethanolamine-N-methyltransferasePhosphatasesPhosphodiesterasesPhosphoinositide-Specific Phospholipase CPhosphoinositide 3-KinasePhospholipase APhospholipase CPhospholipasesPhosphorylasesPhotolysisPI-PLCPI 3-KinasePI 3-Kinase/Akt SignalingPI3KPim-1Pim KinasePIP2Pituitary Adenylate Cyclase Activating Peptide ReceptorsPKAPKBPKCPKDPKG
PKMPLAPlasminPlatelet-Activating Factor (PAF) ReceptorsPlatelet Derived Growth Factor ReceptorsPLCPLKPMCAPNMTPolo-like KinasePoly(ADP-ribose) PolymerasePolyamine OxidasePolyamine SynthasePolymerasesPorcnPost-translational ModificationPotassium (KCa) ChannelsPotassium (KIR) ChannelsPotassium (KV) ChannelsPotassium ChannelsPotassium Channels, Non-SelectivePotassium Channels, OtherPotassium IonophorePPAR, Non-SelectivePPARαPPARδPPARγPPARPregnane X ReceptorsPrion ProteinProgesterone ReceptorsProstacyclinProstaglandinProstanoid ReceptorsProtease-Activated ReceptorsProteasesProteasomeProteinasesProtein Kinase, Broad SpectrumProtein Kinase AProtein Kinase BProtein Kinase CProtein Kinase DProtein Kinase GProtein Ser/Thr PhosphatasesProtein SynthesisProtein Tyrosine PhosphatasesPrP-ResPTH ReceptorsPTPPurinergic (P2Y) ReceptorsPurine TransportersPXRPyrimidine Transporters
S1P ReceptorssAHP ChannelsScreening LibrariesSec7SecretaseSecretase, γ-Secretin ReceptorsSelectinsSensory Neuron-Specific ReceptorsSERCASerine ProteaseSerotonin (5-HT1) ReceptorsSerotonin (5-HT1A) ReceptorsSerotonin (5-HT1B) ReceptorsSerotonin (5-HT1D) ReceptorsSerotonin (5-ht1E) ReceptorsSerotonin (5-HT1F) ReceptorsSerotonin (5-HT2) ReceptorsSerotonin (5-HT2A) ReceptorsSerotonin (5-HT2B) ReceptorsSerotonin (5-HT2C) ReceptorsSerotonin (5-HT3) ReceptorsSerotonin (5-HT4) ReceptorsSerotonin (5-ht5) ReceptorsSerotonin (5-HT6) ReceptorsSerotonin (5-HT7) ReceptorsSerotonin N-acetyl transferaseSerotonin ReceptorsSerotonin RelatedSerotonin TransportersSerotonin UptakeSERTSF-1sGCShp1Shp2Sigma, GeneralSigma-RelatedSigma1 ReceptorsSigma2 Receptors
Sigma ReceptorsSignal Transducers and Activators of TranscriptionSignal TransductionSir2-like Family DeacetylasesSirtuinSmoothened ReceptorsSmo ReceptorsSNSRSOC ChannelsSodium (Epithelial) ChannelsSodium (NaV) ChannelsSodium, Potassium, Chloride CotransporterSodium/Calcium ExchangerSodium ChannelsSomatostatin (sst) ReceptorsSpermidine acetyltransferaseSpermine acetyltransferaseSphingosine-1-Phosphate ReceptorsSphingosine KinaseSphingosine N-acyltransferaseSphKsPLA2Src Kinasesst ReceptorsSTATStem Cell DedifferentiationStem Cell DifferentiationStem Cell ProliferationStem CellsStem Cell SignalingSteroid Hormone ReceptorsSteroidogenic Factor-1STIM-Orai ChannelsSTK-1Store Operated Calcium ChannelsSyk KinaseSynthases, OtherSynthases/SynthetasesSynthetaseSynthetases, Other
T-Type Calcium ChannelsTachykinin, Non-SelectiveTachykinin NK1 ReceptorsTachykinin NK2 ReceptorsTachykinin NK3 ReceptorsTachykinin ReceptorsTankyraseTauTelomeraseTGF-β ReceptorsThrombinThromboxane A2 SynthetaseThromboxane ReceptorsThymidylate SynthetaseThyrotropin-Releasing Hormone ReceptorsTLRTNF-αToll-like ReceptorsTopoisomeraseTP Receptors
Transcription FactorsTransferasesTransforming Growth Factor Beta ReceptorsTransient Receptor Potential ChannelsTranslocation, Exocytosis & EndocytosisTransportersTRH ReceptorsTriphosphoinositol ReceptorsTrk ReceptorsTRPA1TRP ChannelsTRP Channels, OtherTRPMTRPVTrypsinTryptaseTryptophan HydroxylaseTubulinTumor Necrosis Factor-α
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