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Home » Pharmacology » All Targets
All Targets
Pharmacological targets listed alphabetically
κBA1 ReceptorsA2A ReceptorsA2B ReceptorsA3 ReceptorsAbl KinaseACATACEAcetylcholine Muscarinic ReceptorsAcetylcholine Nicotinic ReceptorsAcetylcholine, OtherAcetylcholine α4β2 Nicotinic ReceptorsAcetylcholine α7 Nicotinic ReceptorsAcetylcholine Nicotinic Receptors, Non-selectiveAcetylcholine Nicotinic Receptors, Other SubtypesAcetylcholinesteraseAcetylcholine TransportersAChEAcid sensing ion channel 3ActinActivator Protein-1Activin Receptor-like KinaseAcyl-CoA:cholesterol acyltransferaseacylsphingosine deacylaseAcyltransferasesAdenine ReceptorsAdenosine, OtherAdenosine A1 ReceptorsAdenosine A2A ReceptorsAdenosine A2B ReceptorsAdenosine A3 ReceptorsAdenosine DeaminaseAdenosine KinaseAdenosine ReceptorsAdenosine TransportersAdenosine UptakeAdenylyl CyclaseADKAdrenergic α1 ReceptorsAdrenergic α2 ReceptorsAdrenergic Alpha Receptors, Non-SelectiveAdrenergic β1 ReceptorsAdrenergic β2 ReceptorsAdrenergic β3 ReceptorsAdrenergic Beta Receptors, Non-SelectiveAdrenergic ReceptorsAdrenergic Related CompoundsAdrenergic TransportersAdrenoceptorsAHRAkt (Protein Kinase B)Alcohol DehydrogenaseAldehyde DehydrogenaseAldehyde ReductaseAldose ReductaseAldosterone ReceptorsALK Receptors
Alpha-GlucosidaseAlpha-MannosidaseAlpha4Beta2 Nicotinic ReceptorsAlpha7 Nicotinic ReceptorsAlpha1 Adrenergic ReceptorsAlpha2 Adrenergic ReceptorsAminopeptidaseAMP-Activated Protein KinaseAMPA ReceptorsAMPKAMTAmylin ReceptorsAmyloid β Peptides Amyloid Precursor ProteinAMY ReceptorsAnandamide AmidaseAnandamide TransportersAndrogen ReceptorsAngiogenesisAngiotensin-Converting EnzymeAngiotensin AT1 ReceptorsAngiotensin AT2 ReceptorsAngiotensin ReceptorsAngiotensin Receptors, Non-SelectiveAnkyrin ReceptorsAnnexinANP ReceptorsAntiangiogenicsAntibioticsAntioxidantsAntiprionAntiviralsAP-1Apelin ReceptorAPJ ReceptorApoptosisApoptosis, OtherApoptosis InducersAPP SecretaseAromatic L-Amino Acid DecarboxylaseAryl Hydrocarbon ReceptorsASIC3AT1 ReceptorsAT2 ReceptorsAtaxia Telangiectasia and Rad3 Related KinaseAtaxia Telangiectasia Mutated KinaseATM and ATR KinasesATPaseATPases/GTPasesAT Receptors, Non-SelectiveAtrial Natriuretic Peptide ReceptorsATR KinaseAurora KinaseAutophagyAutotaxinAXOR12 Receptor
c-Ablc-Fosc-IAPc-RafC3Calcium-Activated Potassium (KCa) ChannelsCa2+-ATPaseCaV ChannelsCa2+ Binding Protein ModulatorsCa2+ ChannelsCa2+ IonophoreCa2+Sensitive Protease ModulatorsCa2+ SignalingCa2+ Signaling Agents, GeneralCaged CompoundsCalcineurinCalcitonin and Related ReceptorsCalcium (CaV) ChannelsCalcium-ATPaseCalcium-Sensing ReceptorCalcium-Sensitive Protease ModulatorsCalcium Binding Protein ModulatorsCalcium ChannelsCalcium Channels, OtherCalcium IonophoreCalcium SignalingCalcium Signaling Agents, GeneralCalmodulinCalmodulin-Activated Protein KinaseCalpainsCaM KinaseCaM Kinase KinasecAMPCannabinoid (CB1) ReceptorsCannabinoid (CB2) ReceptorsCannabinoid (GPR55) ReceptorsCannabinoid, Non-SelectiveCannabinoid, OtherCannabinoid ReceptorsCannabinoid TransportersCarbohydrate MetabolismCarbonate dehydrataseCarbonic acid anhydrateCarbonic anhydraseCarbonic AnhydrasesCarboxyanhydrateCarboxypeptidaseCarrier ProteinCasein Kinase 1Casein Kinase 2CaspasesCASRCatecholamine O-methyltransferaseCatechol methyltransferaseCatechol O-MethyltransferaseCatechol O-methyltransferaseCathepsinCB1 ReceptorsCB2 ReceptorsCCK-Inactivating Serine ProteaseCCK1 ReceptorsCCK2 ReceptorsCCK ReceptorsCCR
cdc7Cdc25 PhosphataseCdkCell Adhesion MoleculesCell CycleCell Cycle InhibitorsCell MetabolismCell SignalingCellular ProcessesCeramidaseCeramidasesCeramide-Specific GlycosyltransferaseCFTRCGRP ReceptorsChannel Modulators, OtherCheckpoint Control KinasesCheckpoint KinaseChemokine ReceptorsChk1Chk2Chloride ChannelsCholecystokinin ReceptorsCholecystokinin, Non-SelectiveCholecystokinin1 ReceptorsCholecystokinin2 ReceptorsCholinesterasesChymaseCK1CK2Cl- ChannelsClassical ReceptorscMETComplementCOMTConnexinsConvertase, C3-Corticotropin-Releasing Factor, Non-SelectiveCorticotropin-Releasing Factor1 ReceptorsCorticotropin-Releasing Factor2 ReceptorsCorticotropin-Releasing Factor ReceptorsCOXCRF, Non-SelectiveCRF1 ReceptorsCRF2 ReceptorsCRF ReceptorsCRTH2CT ReceptorsCXCRCyclasesCyclic Adenosine MonophosphateCyclic Nucleotide Dependent-Protein KinaseCyclin-Dependent Protein KinaseCyclooxygenaseCYPCysLT1 ReceptorsCysLT2 ReceptorsCysteinyl Aspartate ProteaseCytidine DeaminaseCytochrome P450Cytokine and NF-κB SignalingCytokine ReceptorsCytokinesCytoskeleton & Motor Proteins
D1 and D5 ReceptorsD2 ReceptorsD3 ReceptorsD4 ReceptorsDAG KinaseDAGLDAPKDardarinDATDeacetylasesDeaminasesDeath Domain Receptor-Associated Adaptor KinaseDecarboxylasesDehydrogenasesΔ7-Dehydrocholesterol ReductaseDelta Opioid ReceptorsDemethylasesDeoxycytidine KinaseDGAT-1DGKDHCRDHFRDiacylglycerolacyltransferase 1Diacylglycerol KinaseDiacylglycerol LipaseDihydrofolate ReductaseDihydrotestosterone Receptors
DipeptidaseDipeptidyl Peptidase IVDMTasesDMTsDNA, RNA and Protein SynthesisDNA-Dependent Protein KinaseDNA-PKDNA LigaseDNA LigasesDNA MethyltransferasesDNA TopoisomeraseDNMTsDopamine D1 ReceptorsDopamine D2-like, Non-SelectiveDopamine D2 ReceptorsDopamine D3 ReceptorsDopamine D4 ReceptorsDopamine D5 ReceptorsDopamine ReceptorsDopaminergic-RelatedDopamine TransportersDOP ReceptorsDPP-IVDP ReceptorsDual-Specificity PhosphataseDynamin
E-Type ATPaseEAATECEEcto-ATPaseEDG ReceptorsEGFRElastaseElk3ENaCEncephalitogenic Myelin Oligodendrocyte GlycoproteinEncephalitogenic Myelin Proteolipid FragmentEndocytosisEndopeptidase 24.15Endothelial LipaseEndothelial Nitric Oxide SynthaseEndothelin, Non-SelectiveEndothelin-Converting EnzymeETA ReceptorsETB ReceptorsEndothelin ReceptorseNOSENPP2ENT1Enzyme-Associated ReceptorsEnzyme-Linked ReceptorsEnzymesEnzyme Substrates / Activators
EP1-4 ReceptorsEpacEpidermal Growth Factor ReceptorsEpigenetic erasersEpigenetic readersEpigeneticsEpigenetic writersEpithelial Sodium ChannelsEquilibrative Nucleoside TransportersERErbBERKERRE SelectinEsterasesEstrogen (GPR30) ReceptorsEstrogen ReceptorsET, Non-SelectiveETA ReceptorsETB ReceptorsET ReceptorsExcitatory Amino Acid TransportersExocytosisExonucleasesExtracellular Matrix and Adhesion MoleculesExtracellular Signal-Regulated Kinase
G-Protein-Coupled ReceptorsGβγGi/oGq/11GsGABA, MiscellaneousGABA-TransferaseGABAA and GABAC ReceptorsGABAA ReceptorsGABAB ReceptorsGABAC ReceptorsGABA TransportersGalanin ReceptorsGAL ReceptorsGamma-SecretaseGap ChannelsGastric Inhibitory Polypeptide ReceptorGastrin-Releasing Peptide-Preferring ReceptorsGATGCPGeneral Calcium Signaling AgentsGeneral ImidazolinesGeranylgeranyltransferaseGhrelin ReceptorsGHS-R1a ReceptorsGIP ReceptorGLASTGLP1 ReceptorsGLP2 ReceptorsGLT-1Glucagon-Like Peptide 1 ReceptorsGlucagon-Like Peptide 2 ReceptorsGlucagon and Related ReceptorsGlucagon ReceptorGlucocorticoid ReceptorsGlucose-Dependent Insulinotropic PeptideGlucose TransportersGlucosidaseGLUTGlutamate (AMPA) Receptors
Glutamate (Ionotropic), Non-SelectiveGlutamate (Ionotropic) ReceptorsGlutamate (Kainate) ReceptorsGlutamate (Metabotropic) Group III ReceptorsGlutamate (Metabotropic) Group II ReceptorsGlutamate (Metabotropic) Group I ReceptorsGlutamate (Metabotropic) ReceptorsGlutamate (NMDA) ReceptorsGlutamate, MiscellaneousGlutamate Carboxypeptidase IIGlutamate (EAAT) TransportersGlutathione S-TransferaseGlycine ReceptorsGlycine TransportersGlycogen PhosphorylaseGlycogen Synthase Kinase 3Glycoprotein IIb/IIIa (αIIbα3)glycosphingolipid ceramide deacylaseGlycosylasesGlycosyltransferaseGlyRGlyTGnRH ReceptorsGonadotropin-Releasing Hormone ReceptorsGPCRGPR30 ReceptorsGPR35GPR40 ReceptorsGPR54 ReceptorGPR55GPR119GPR119 GPR_119G Proteins (Heterotrimeric)G Proteins (Small)Growth Factor ReceptorsGrowth Hormone Secretagog Receptor 1aGRP-Preferring ReceptorsGSKGTPaseGuanylyl Cyclase
H+, K+-ATPaseH+-ATPaseH1 ReceptorsH2 ReceptorsH3 ReceptorsH4 ReceptorsHATsHDACsHeat Shock Protein 70Heat Shock Protein 90Heat Shock ProteinsHedgehog SignalingHeme OxygenaseHeparanaseHepatocyte Growth Factor ReceptorsHerhERG ChannelsHexokinaseHexosaminidase, BetaHGFRHh SignalingHIFHistamine H1 ReceptorsHistamine H2 ReceptorsHistamine H3 ReceptorsHistamine H4 Receptors
Histamine ReceptorsHistaminergic-Related CompoundsHistone AcetyltransferasesHistone DeacetylasesHistone DemethylasesHistone MethyltransferasesHMG-CoA ReductaseHormone-sensitive LipasehOT7T175 ReceptorHSLHsp70Hsp90HspsHuman Ether-A-Go-Go Related Gene ChannelsHuman Leukocyte ElastaseHuman Neutrophil ElastaseHydrogen, Potassium-ATPaseHydrogen-ATPaseHydrolasesHydroxycarboxylic Acid ReceptorsHydroxylase, 11-βHydroxylasesHydroxysteroid Dehydrogenase, 11β-Hydroxytryptamine, 5- ReceptorsHydroxytryptamine, 5- Transporters
I1 ReceptorsI2 ReceptorsI3 ReceptorsIAPICAMIGF ReceptorsiGlu ReceptorsIκB KinaseIKKIL ReceptorsImidazoline (I1) ReceptorsImidazoline (I2) ReceptorsImidazoline (I3) ReceptorsImidazoline, GeneralImidazoline ReceptorsImmunosuppressantsIMPaseInducible Nitric Oxide SynthaseInhibitor of ApoptosisInhibitor of Kappa BiNOSInositol 1,4,5-triphosphate Receptors
Inositol and cAMP SignalingInositol LipidsInositol MonophosphataseInositol PhosphatasesIns(1,4,5)P3 5-PhosphataseInsulin and Insulin-like ReceptorsIntegrin ReceptorsInterleukin ReceptorsInterleukinsInward Rectifier Potassium (Kir) ChannelsIon ChannelsIonophoresIonotropic Glutamate ReceptorsIon Pumps, OtherIon Pumps/TransportersIon TransportersIon Transporters, OtherIP3 ReceptorsIP ReceptorsIRE1Isomerases
M1 ReceptorsM2 ReceptorsM3 ReceptorsM4 ReceptorsM5 ReceptorsMAGLMammalian Target of RapamycinMannosidaseMAOMAPKMAPK, OtherMAPK SignalingMatrixinsMatrix MetalloproteaseMatrix Metalloproteinase (MMP)Maxi-K ChannelsMBOATMCH ReceptorsMcl-1MC ReceptorsMCUMDM2MDRMEKMelanin-concentrating Hormone ReceptorsMelanocortin (MC) ReceptorsMelastatin ReceptorsMelatonin ReceptorsMembrane-bound O-acyltransferase (MBOAT)Membrane Transport ProteinMET ReceptorMetabotropic Glutamate ReceptorsMetastin ReceptorMethionine Aminopeptidase-2mGlu, Non-SelectivemGlu1 ReceptorsmGlu2 ReceptorsmGlu3 ReceptorsmGlu4 ReceptorsmGlu5 ReceptorsmGlu6 ReceptorsmGlu7 ReceptorsmGlu8 Receptors
mGlu Group III ReceptorsmGlu Group II ReceptorsmGlu Group I ReceptorsmGlu ReceptorsMicrotubulesMineralocorticoid ReceptorsMiscellaneous OpioidsMiscellaneous CompoundsMiscellaneous GABAMiscellaneous GlutamateMitochondrial Calcium UniporterMitochondrial HexokinaseMitogen-Activated Protein KinaseMitogen-Activated Protein Kinase-Activated Protein Kinase-2Mitogen-Activated Protein Kinase KinaseMitosisMitotic Kinesin Eg5MK-2MLCKMMPMnk1Monoacylglycerol LipaseMonoamine OxidaseMonoamine TransportersMOP ReceptorsMotilin ReceptorMotor ProteinsMPTPMre11-Rad50-Nbs1MRN ExonucleasemTORMT ReceptorsMucolipin ReceptorsMultidrug TransportersMu Opioid ReceptorsMuscarinic (M1) ReceptorsMuscarinic (M2) ReceptorsMuscarinic (M3) ReceptorsMuscarinic (M4) ReceptorsMuscarinic (M5) ReceptorsMuscarinic ReceptorsMyosinMyosin Light Chain Kinase
N-Methyl-D-Aspartate ReceptorsN-Myristoyltransferase-1N-Type Calcium ChannelsNa+/Ca2+ ExchangerNa+/H+ ExchangerNa+/K+ ATPaseNaV ChannelsNa+/2Cl-/K+ CotransporterNa+ ChannelsNAAG PeptidaseNAALADasenAChRNADPH OxidaseNatriuretic Peptide ReceptorsNCAMNCXNeovascularizationNETNetNeurokinin ReceptorsNeurolysinNeuromedin B-Preferring ReceptorsNeuromedin U ReceptorsNeuronal MetabolismNeuronal Nitric Oxide SynthaseNeuropeptide FF/AF ReceptorsNeuropeptide Y ReceptorsNeurotensin ReceptorsNeurotransmitter TransportersNeurotrophin ReceptorsNeutrophil ElastaseNF-κB & IκBNFE2L2NHENicotinic (α4β2) ReceptorsNicotinic (α7) ReceptorsNicotinic Acid ReceptorsNicotinic ReceptorsNicotinic Receptors (Non-selective)Nicotinic Receptors (Other Subtypes)Nitric Oxide, OtherNitric Oxide DonorsNitric Oxide PrecursorsNitric Oxide SignalingNitric Oxide SynthaseNitric Oxide Synthase, Non-SelectiveNK1 ReceptorsNK2 Receptors
NK3 ReceptorsNKCC CotransporterNMB-Preferring ReceptorsNMDA ReceptorsNME2NMU ReceptorsnNOSNociceptin ReceptorsNO Donors / PrecursorsNogo-66 ReceptorsNon-selective / Other Potassium ChannelsNon-selective 5-HTNon-selective 5-HT1Non-selective 5-HT2Non-selective AdenosineNon-selective Adrenergic α ReceptorsNon-selective Adrenergic β ReceptorsNon-selective AT ReceptorsNon-selective CannabinoidsNon-selective CCKNon-selective CRFNon-selective DopamineNon-selective EndothelinNon-selective Ionotropic GlutamateNon-selective Metabotropic GlutamateNon-selective MuscarinicsNon-selective NOSNon-selective OrexinNon-selective PPARNon-selective TRP ChannelsNOP ReceptorsNO PrecursorsNoradrenalin TransporterNO Synthase, Non-SelectiveNO SynthasesNotch SignalingNOXNPFF ReceptorsNPP2NPRNPY ReceptorsNrf2NTPDaseNT ReceptorsNuclear Factor Kappa BNuclear ReceptorsNuclear Receptors, OtherNucleoside Transporters
O-GlcNAcaseOATP1B1OP1 ReceptorsOP2 ReceptorsOP3 ReceptorsOP4 ReceptorsOpioid, δ-Opioid, κ-Opioid, μ-Opioid ReceptorsOrexin, Non-SelectiveOrexin1 ReceptorsOrexin2 ReceptorsOrexin ReceptorsOrganic Anion Transporting PolypeptideORL1 ReceptorsOrnithine DecarboxylaseOrphan 7-TM ReceptorsOrphan 7-Transmembrane ReceptorsOrphan G-Protein-Coupled ReceptorsOrphan GPCRsOther AcetylcholineOther AdenosineOther ApoptosisOther ATPasesOther Calcium ChannelsOther CannabinoidsOther Channel ModulatorsOther Dehydrogenases
Other EpigeneticsOther HydrolasesOther Ion Pumps/TransportersOther KinasesOther MAPKOther Nitric OxideOther Nuclear ReceptorsOther Oxygenases/OxidasesOther Peptide ReceptorsOther PharmacologyOther Product TypesOther ProteasesOther ReductasesOther RTKsOther Synthases/SynthetasesOther TachykininOther Transcription FactorsOther TransferasesOther Wnt SignalingOT ReceptorsOX1 ReceptorsOX2 ReceptorsOXE ReceptorsOxidaseOxidative PhosphorylationOxoeicosanoid receptorsOxygenases/OxidasesOxytocin Receptors
P-GlycoproteinP-SelectinP-Type ATPaseP-Type Calcium ChannelsP2X ReceptorsP2Y Receptorsp14ARFp38 MAPKp53p56lckp60c-srcp70 S6Kp75p90 Ribosomal S6 Kinasep160ROCKPAC1 ReceptorsPACAP ReceptorsPAF ReceptorsPAOParathyroid Hormone ReceptorsPARPPAR ReceptorsPC-PLCPDEPDGFRPDK1PDPK1Peptide Receptor, OtherPeptide ReceptorsPeroxisome-Proliferating ReceptorsPGFPGI2PhosphatasesPhosphodiesterasesPhosphoinositide-Specific Phospholipase CPhosphoinositide 3-KinasePhospholipase APhospholipase CPhospholipasesPhosphorylasesPhotolysisPI-PLCPI 3-KinasePI 3-Kinase/Akt SignalingPI3KPim-1Pim KinasePIP2Pituitary Adenylate Cyclase Activating Peptide ReceptorsPKAPKBPKCPKDPKGPKMPKMTs
PLAPlasminPlatelet-Activating Factor (PAF) ReceptorsPlatelet Derived Growth Factor ReceptorsPLCPLKPMCAPolo-like KinasePoly(ADP-ribose) PolymerasePolyamine OxidasePolyamine SynthasePolycystin ReceptorsPolymerasesPorcnPost-translational ModificationPotassium (KCa) ChannelsPotassium (Kir) ChannelsPotassium (KV) ChannelsPotassium ChannelsPotassium Channels, Non-selectivePotassium Channels, OtherPotassium IonophorePPAR, Non-SelectivePPARαPPARδPPARγPPARPregnane X ReceptorsPrion ProteinPRMTsProgesterone ReceptorsProstacyclinProstaglandinProstanoid ReceptorsProtease-Activated ReceptorsProteasesProteasomeProteinasesProtein Kinase, Broad SpectrumProtein Kinase AProtein Kinase BProtein Kinase CProtein Kinase DProtein Kinase GProtein MethyltransferasesProtein Ser/Thr PhosphatasesProtein SynthesisProtein Tyrosine PhosphatasesPrP-ResPTH ReceptorsPTPPurinergic P1 ReceptorsPurinergic (P2Y) ReceptorsPurine TransportersPXRPyrimidine Transporters
S1P ReceptorssAHP ChannelsScreening LibrariesSec7Secretin ReceptorsSelectinsSensory Neuron-Specific ReceptorsSERCASerine ProteaseSerotonin (5-HT1) ReceptorsSerotonin (5-HT1A) ReceptorsSerotonin (5-HT1B) ReceptorsSerotonin (5-HT1D) ReceptorsSerotonin (5-ht1E) ReceptorsSerotonin (5-HT1F) ReceptorsSerotonin (5-HT2) ReceptorsSerotonin (5-HT2A) ReceptorsSerotonin (5-HT2B) ReceptorsSerotonin (5-HT2C) ReceptorsSerotonin (5-HT3) ReceptorsSerotonin (5-HT4) ReceptorsSerotonin (5-ht5) ReceptorsSerotonin (5-HT6) ReceptorsSerotonin (5-HT7) ReceptorsSerotonin N-acetyl transferaseSerotonin ReceptorsSerotonin RelatedSerotonin TransportersSerotonin UptakeSERTSF-1sGCShp1Shp2Sigma, GeneralSigma-RelatedSigma1 ReceptorsSigma2 ReceptorsSigma ReceptorsSignal Transducers and Activators of Transcription
Signal TransductionSir2-like Family DeacetylasesSirtuinSmoothened ReceptorsSmo ReceptorsSNSRSOC ChannelsSodium (Epithelial) ChannelsSodium (NaV) ChannelsSodium, Potassium, Chloride CotransporterSodium/Calcium ExchangerSodium/Hydrogen ExchangerSodium ChannelsSomatostatin (sst) ReceptorsSpermidine acetyltransferaseSpermine acetyltransferaseSphingosine-1-Phosphate ReceptorsSphingosine KinaseSphingosine N-acyltransferaseSphKsPLA2Src Kinasesst ReceptorsSTATStem Cell DedifferentiationStem Cell DifferentiationStem Cell ProliferationStem CellsStem Cell SignalingSteroid Hormone ReceptorsSteroidogenic Factor-1STIM-Orai ChannelsSTK-1Store Operated Calcium ChannelsSyk KinaseSynthases, OtherSynthases/SynthetasesSynthetaseSynthetases, Other
T-Type Calcium ChannelsTachykinin, Non-SelectiveTachykinin NK1 ReceptorsTachykinin NK2 ReceptorsTachykinin NK3 ReceptorsTachykinin ReceptorsTankyraseTauTelomeraseTGF-β ReceptorsThrombinThromboxane A2 SynthetaseThromboxane ReceptorsThymidylate SynthetaseThyrotropin-Releasing Hormone ReceptorsTLRTNF-αToll-like ReceptorsTopoisomeraseTP ReceptorsTranscription FactorsTransferasesTransforming Growth Factor Beta Receptors
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