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Home » Pharmacology » All Targets
All Targets
Pharmacological targets listed alphabetically
A1 ReceptorsA2A ReceptorsA2B ReceptorsA3 ReceptorsAbl KinaseACATACEAcetylcholine Muscarinic ReceptorsAcetylcholine Nicotinic ReceptorsAcetylcholine, OtherAcetylcholine α4β2 Nicotinic ReceptorsAcetylcholine α7 Nicotinic ReceptorsAcetylcholine Nicotinic Receptors, Non-SelectiveAcetylcholine Nicotinic Receptors, Other SubtypesAcetylcholinesteraseAcetylcholine TransportersAChEAcid sensing ion channel 3ActinActivator Protein-1Activin Receptor-like KinaseAcyl-CoA:cholesterol acyltransferaseAcyltransferasesAdenosine, OtherAdenosine A1 ReceptorsAdenosine A2A ReceptorsAdenosine A2B ReceptorsAdenosine A3 ReceptorsAdenosine DeaminaseAdenosine KinaseAdenosine ReceptorsAdenosine TransportersAdenosine UptakeAdenylyl CyclaseAdhesion MoleculesADKAdrenergic α1 ReceptorsAdrenergic α2 ReceptorsAdrenergic Alpha Receptors, Non-SelectiveAdrenergic β1 ReceptorsAdrenergic β2 ReceptorsAdrenergic β3 ReceptorsAdrenergic Beta Receptors, Non-SelectiveAdrenergic ReceptorsAdrenergic Related CompoundsAdrenergic TransportersAdrenoceptorsAHRAkt (Protein Kinase B)Alcohol Dehydrogenase 7Aldehyde ReductaseAldose ReductaseAldosterone ReceptorsALK Receptors
Alpha-GlucosidaseAlpha-MannosidaseAlpha4Beta2 Nicotinic ReceptorsAlpha7 Nicotinic ReceptorsAlpha1 Adrenergic ReceptorsAlpha2 Adrenergic ReceptorsAminopeptidaseAMP-Activated Protein KinaseAMPA ReceptorsAMPKAMTAmylin ReceptorsAmyloid β Peptides Amyloid Precursor ProteinAMY ReceptorsAnandamide AmidaseAnandamide TransportersAndrogen ReceptorsAngiogenesisAngiotensin-Converting EnzymeAngiotensin AT1 ReceptorsAngiotensin AT2 ReceptorsAngiotensin AT4 ReceptorsAngiotensin ReceptorsAngiotensin Receptors, Non-SelectiveAnnexinANP ReceptorsAntiangiogenicsAntibodiesAntiprion AP-1Apelin ReceptorsAPJ ReceptorsApoptosisApoptosis, OtherApoptosis InducerAPP SecretaseAromatic L-Amino Acid DecarboxylaseAryl Hydrocarbon ReceptorsASIC3AT1 ReceptorsAT2 ReceptorsAT4 ReceptorsAtaxia Telangiectasia and Rad3 Related KinaseAtaxia Telangiectasia Mutated KinaseATM and ATR KinasesATPaseATPases/GTPasesAT Receptors, Non-SelectiveAtrial Natriuretic Peptide ReceptorsATR KinaseAurora KinaseAXOR12 Receptors
c-Ablc-Fosc-IAPc-Junc-Jun N-Terminal Kinasec-RafC3Ca2+-Activated Potassium (KCa) ChannelsCa2+-ATPaseCaV ChannelsCa2+ Binding Protein ModulatorsCa2+ ChannelsCa2+ IonophoreCa2+Sensitive Protease ModulatorsCa2+ SignalingCa2+ Signaling Agents, GeneralCaged CompoundsCalcineurinCalcitonin and Related ReceptorsCalcium (CaV) ChannelsCalcium-ATPaseCalcium-Sensitive Protease ModulatorsCalcium Binding Protein ModulatorsCalcium ChannelsCalcium Channels, OtherCalcium IonophoreCalcium SignalingCalcium Signaling Agents, GeneralCalmodulinCalmodulin-Activated Protein KinaseCalpainCaM KinaseCaM Kinase KinasecAMPCannabinoid (CB1) ReceptorsCannabinoid (CB2) ReceptorsCannabinoid (GPR55) ReceptorsCannabinoid, Non-SelectiveCannabinoid, OtherCannabinoid ReceptorsCannabinoid TransportersCarbohydrate MetabolismCarboxypeptidaseCarrier ProteinCasein Kinase 1Casein Kinase 2CaspaseCatechol-O-methyltransferaseCathepsinCB1 ReceptorsCB2 ReceptorsCCK-Inactivating Serine ProteaseCCK1 ReceptorsCCK2 ReceptorsCCK ReceptorsCCRcdc7
Cdc25 PhosphataseCdkCell CycleCell Cycle InhibitorsCell MetabolismCell SignalingCellular ProcessesCeramidaseCeramide-Specific GlycosyltransferaseCFTRCGRP ReceptorsChannel Modulators, OtherCheckpoint Control KinasesCheckpoint KinaseChemokine ReceptorsChk1Chk2Chloride ChannelsCholecystokinin ReceptorsCholecystokinin, Non-SelectiveCholecystokinin1 ReceptorsCholecystokinin2 ReceptorsCholinesteraseCK1CK2Cl- ChannelscMETComplementCOMTConnexinsConvertase, C3-Corticotropin-Releasing Factor, Non-SelectiveCorticotropin-Releasing Factor1 ReceptorsCorticotropin-Releasing Factor2 ReceptorsCorticotropin-Releasing Factor ReceptorsCOXCRF, Non-SelectiveCRF1 ReceptorsCRF2 ReceptorsCRF ReceptorsCRTH2CT ReceptorsCXCRCyclasesCyclic Adenosine MonophosphateCyclic Nucleotide Dependent-Protein KinaseCyclin-Dependent Protein KinaseCyclooxygenaseCYPCysLT1 ReceptorsCysLT2 ReceptorsCytidine DeaminaseCytochrome P450Cytokine and NF-κB SignalingCytokine ReceptorsCytokinesCytoskeleton & Motor Proteins
D1 and D5 ReceptorsD2 ReceptorsD3 ReceptorsD4 ReceptorsDAG KinaseDAGLDATDeacetylasesDeaminasesDeath Domain Receptor-Associated Adaptor KinaseDecarboxylasesDehydrogenasesΔ7-Dehydrocholesterol Reductaseδ Opioid ReceptorsDeoxycytidine KinaseDGKDHCRDHFRDiacylglycerol KinaseDiacylglycerol LipaseDihydrofolate ReductaseDihydroorotate DehydrogenaseDihydrotestosterone Receptors
DipeptidaseDipeptidyl Peptidase IVDNA, RNA and Protein SynthesisDNA-Dependent Protein KinaseDNA-PKDNA LigaseDNA methyltransferaseDNA TopoisomeraseDopamine D1 ReceptorsDopamine D2-like, Non-SelectiveDopamine D2 ReceptorsDopamine D3 ReceptorsDopamine D4 ReceptorsDopamine D5 ReceptorsDopamine ReceptorsDopaminergic-RelatedDopamine TransportersDOP ReceptorsDPP-IVDP ReceptorsDual-Specificity PhosphataseDynamin
E-Type ATPaseEAATECEEDG ReceptorsEGFRElastaseElk3ENaCEncephalitogenic Myelin Oligodendrocyte GlycoproteinEncephalitogenic Myelin Proteolipid FragmentEndocytosisEndopeptidase 24.15Endothelial Nitric Oxide SynthaseEndothelin, Non-SelectiveEndothelin-Converting EnzymeETA ReceptorsETB ReceptorsEndothelin ReceptorseNOSENT1Enzyme-Associated ReceptorsEnzyme-Linked Receptors
EnzymesEnzyme Substrates / ActivatorsEP1-4 ReceptorsEpacEpidermal Growth Factor ReceptorsEpithelial Sodium ChannelsEquilibrative Nucleoside TransportersERErbBERRE SelectinEsterasesEstrogen (GPR30) ReceptorsEstrogen ReceptorsET, Non-SelectiveETA ReceptorsETB ReceptorsET ReceptorsExcitatory Amino Acid TransportersExocytosisExonucleaseExtracellular Matrix and Adhesion Molecules
G-Protein-Coupled ReceptorsGβγGi/oGq/11GsGABA, MiscellaneousGABA-TransferaseGABAA and GABAC ReceptorsGABAA ReceptorsGABAB ReceptorsGABAC ReceptorsGABA TransportersGalanin ReceptorsGAL ReceptorsGamma-SecretaseGap ChannelsGastric Inhibitory Peptide ReceptorsGastrin-Releasing Peptide-Preferring ReceptorsGATGCPGeneral Calcium Signaling AgentsGeneral ImidazolinesGeneral SigmaGeranylgeranyltransferaseGhrelin ReceptorsGHRH ReceptorsGHS-R1a ReceptorsGIP ReceptorsGLASTGLP1 ReceptorsGLP2 ReceptorsGLT-1Glucagon-Like Peptide 1 ReceptorsGlucagon-Like Peptide 2 ReceptorsGlucagon and Related ReceptorsGlucagon ReceptorsGlucocorticoid ReceptorsGlucose-Dependent Insulinotropic PeptideGlucosidase
Glutamate (AMPA) ReceptorsGlutamate (Ionotropic), Non-SelectiveGlutamate (Ionotropic) ReceptorsGlutamate (Kainate) ReceptorsGlutamate (Metabotropic) Group III ReceptorsGlutamate (Metabotropic) Group II ReceptorsGlutamate (Metabotropic) Group I ReceptorsGlutamate (Metabotropic) ReceptorsGlutamate (NMDA) ReceptorsGlutamate, MiscellaneousGlutamate Carboxypeptidase IIGlutamate (EAAT) TransportersGlutathione S-TransferaseGlycine ReceptorsGlycine TransportersGlycogen Synthase Kinase 3Glycoprotein IIb/IIIa (αIIbα3)GlycosylasesGlyRGlyTGnRH ReceptorsGonadotrophin-Releasing Hormone ReceptorsGPCRGPR30 ReceptorsGPR40 ReceptorsGPR54 ReceptorsGPR55 ReceptorsGPR109 ReceptorsGPR119 ReceptorsG Proteins (Heterotrimeric)G Proteins (Small)GRF ReceptorsGrowth-Hormone Releasing Hormone ReceptorsGrowth Hormone Secretagog Receptor 1aGRP-Preferring ReceptorsGSKGTPaseGuanylyl Cyclase
H+, K+-ATPaseH+-ATPaseH1 ReceptorsH2 ReceptorsH3 ReceptorsH4 ReceptorsHDACHeat Shock Protein 90Hedgehog SignalingHeme OxygenaseHeparanaseHepatocyte Growth Factor ReceptorsHerhERG ChannelsHexokinaseHexosaminidase, BetaHGFRHh SignalingHistamine H1 ReceptorsHistamine H2 ReceptorsHistamine H3 ReceptorsHistamine H4 Receptors
Histamine N-methyltransferaseHistamine ReceptorsHistaminergic-Related CompoundsHistone DeacetylaseHM74 ReceptorsHMG-CoA ReductaseHormone-sensitive LipasehOT7T175 ReceptorsHSLHsp90Human Ether-A-Go-Go Related Gene ChannelsHuman Leukocyte ElastaseHuman Neutrophil ElastaseHydrogen, Potassium-ATPaseHydrogen-ATPaseHydrolasesHydroxylase, 11-βHydroxylasesHydroxysteroid Dehydrogenase, 11β-Hydroxytryptamine, 5- ReceptorsHydroxytryptamine, 5- Transporters
I1 ReceptorsI2 ReceptorsI3 ReceptorsIκBIAPICAMIGF ReceptorsiGlu ReceptorsIκB KinaseIKKIL ReceptorsImidazoline (I1) ReceptorsImidazoline (I2) ReceptorsImidazoline (I3) ReceptorsImidazoline, GeneralImidazoline ReceptorsIMPaseInducible Nitric Oxide SynthaseInhibitor of ApoptosisInhibitor of Kappa BiNOS
Inositol 1,4,5-triphosphate ReceptorsInositol and cAMP SignalingInositol LipidsInositol MonophosphataseInositol PhosphataseIns(1,4,5)P3 5-PhosphataseInsulin and Insulin-like ReceptorsIntegrin ReceptorsInterleukin ReceptorsInterleukinsInward Rectifier Potassium (KIR) ChannelsIon ChannelsIonophoresIonotropic Glutamate ReceptorsIon Pumps, OtherIon Pumps/TransportersIon TransportersIon Transporters, OtherIP3 ReceptorsIP ReceptorsIsomerases
MAGLMammalian Target of RapamycinMannosidaseMAOMAPKMAPK SignalingMatrixinsMatrix Metalloprotease (MMP)Matrix Metalloproteinase (MMP)Maxi-K ChannelsMCH ReceptorsMcl-1MC ReceptorsMDM2MDRMEKMelanin-Concentrating Hormone ReceptorsMelanocortin (MC) ReceptorsMelatonin ReceptorsMembrane Transport ProteinMET ReceptorsMetabotropic Glutamate ReceptorsMetastin ReceptorsMethionine Aminopeptidase-2MethyltransferasesmGlu, Non-SelectivemGlu1 ReceptorsmGlu2 ReceptorsmGlu3 ReceptorsmGlu4 ReceptorsmGlu5 ReceptorsmGlu6 ReceptorsmGlu7 ReceptorsmGlu8 ReceptorsmGlu Group III ReceptorsmGlu Group II Receptors
mGlu Group I ReceptorsmGlu ReceptorsMicrotubulesMineralocorticoid ReceptorsMiscellaneous OpioidsMiscellaneous CompoundsMiscellaneous GABAMiscellaneous GlutamateMitochondrial HexokinaseMitogen-Activated Protein KinaseMitogen-Activated Protein Kinase-Activated Protein Kinase-2Mitogen-Activated Protein Kinase KinaseMitosisMitotic Kinesin Eg5 MK-2MLCKMMPMnk1Monoacylglycerol LipaseMonoamine OxidaseMonoamine TransportersMonophosphatase DehydrogenaseMOP ReceptorsMotilin ReceptorsMotor ProteinsMre11-Rad50-Nbs1MRN ExonucleasemTORMT ReceptorsMultidrug Transportersμ Opioid ReceptorsMuscarinic ReceptorsMYCMyosin Light Chain KinaseMyosin
N-Methyl-D-Aspartate ReceptorsN-Myristoyltransferase-1N-Type Calcium ChannelsNa+/Ca2+ ExchangerNaV ChannelsNa+/2Cl-/K+ CotransporterNa+ ChannelsNAAG PeptidaseNAALADasenAChRNatriuretic Peptide ReceptorsNCAMNetNETNeurokinin ReceptorsNeurolysinNeuromedin B-Preferring ReceptorsNeuromedin U ReceptorsNeuronal MetabolismNeuronal Nitric Oxide SynthaseNeuropeptide FF/AF ReceptorsNeuropeptide Y ReceptorsNeurotensin ReceptorsNeurotransmitter TransportersNeurotrophin ReceptorsNeutrophil ElastaseNF-κB & IκBNHE-1Nicotinic (α4β2) ReceptorsNicotinic (α7) ReceptorsNicotinic Acid ReceptorsNicotinic ReceptorsNicotinic Receptors (Non-Selective)Nicotinic Receptors (Other Subtypes)Nitric Oxide, OtherNitric Oxide DonorsNitric Oxide PrecursorsNitric Oxide SignalingNitric Oxide SynthaseNitric Oxide Synthase, Non-SelectiveNK1 ReceptorsNK2 Receptors
NK3 ReceptorsNKCC CotransporterNMB-Preferring ReceptorsNMDA ReceptorsNME2NMU ReceptorsnNOSNociceptin ReceptorsNO Donors / PrecursorsNogo-66 ReceptorsNon-Selective / Other Potassium ChannelsNon-selective 5-HTNon-selective 5-HT1Non-selective 5-HT2Non-selective AdenosineNon-selective Adrenergic α ReceptorsNon-selective Adrenergic β ReceptorsNon-selective AT ReceptorsNon-selective CannabinoidsNon-selective CCKNon-selective CRFNon-selective DopamineNon-selective EndothelinNon-Selective Ionotropic GlutamateNon-selective mGluNon-Selective NOSNon-selective OXNon-selective PPARNOP ReceptorsNO PrecursorsNoradrenalin TransporterNO Synthase, Non-SelectiveNO SynthasesNPFF ReceptorsNPRNPY ReceptorsNT ReceptorsNuclear Factor Kappa BNuclear ReceptorsNuclear Receptors, OtherNucleoside Transporters
O-GlcNAcaseOATP1B1OP1 ReceptorsOP2 ReceptorsOP3 ReceptorsOP4 ReceptorsOpioid, δ-Opioid, κ-Opioid, μ-Opioid ReceptorsOrexin, Non-SelectiveOrexin1 ReceptorsOrexin2 ReceptorsOrexin ReceptorsOrganic Anion Transporting PolypeptideORL1 ReceptorsOrnithine DecarboxylaseOther AcetylcholineOther Activin ReceptorsOther AdenosineOther ApoptosisOther Calcium ChannelsOther CannabinoidsOther Channel ModulatorsOther HydrolasesOther Ion Pumps/Transporters
Other KinasesOther Nitric OxideOther Nuclear ReceptorsOther Oxygenases/OxidasesOther Peptide ReceptorsOther PharmacologyOther Product TypesOther ProteasesOther ReductasesOther RTKsOther Synthases/SynthetasesOther TachykininOther Transcription FactorsOther TransferasesOther TRP ChannelsOther Wnt SignalingOT ReceptorsOX1 ReceptorsOX2 ReceptorsOXE ReceptorsOxidaseOxidative phosphorylationOxoeicosanoid receptorsOxygenases/OxidasesOxytocin Receptors
P-GlycoproteinP-SelectinP-Type ATPaseP-Type Calcium ChannelsP2X ReceptorsP2Y Receptorsp14ARFp38 MAPKp53p56lckp60c-srcp75p90 Ribosomal S6 Kinasep90 RSKp160ROCKPAC1 ReceptorsPACAP ReceptorsPAF ReceptorsParathyroid Hormone ReceptorsPARPPAR ReceptorsPC-PLCPDEPDGFRPeptide Receptor, OtherPeptide ReceptorsPeroxisome-Proliferating ReceptorsPGFPGI2PhosphatasesPhosphodiesterasesPhosphoinositide-Specific Phospholipase CPhosphoinositide 3-KinasePhospholipasePhospholipase APhospholipase CPhotolysisPI-PLCPI 3-KinasePI 3-Kinase/Akt SignalingPI3KPim-1Pim-1 KinasePIP2Pituitary Adenylate Cyclase Activating Peptide ReceptorsPKAPKBPKCPKDPKGPKM
PLAPlasminPlatelet-Activating Factor (PAF) ReceptorsPlatelet Derived Growth Factor ReceptorsPLCPLKPMCAPolo-like KinasePoly(ADP-ribose) PolymerasePolyamine OxidasePolyamine SynthasePolymerasesPost-translational ModificationPotassium (KCa) ChannelsPotassium (KIR) ChannelsPotassium (KV) ChannelsPotassium ChannelsPotassium Channels, Non-SelectivePotassium Channels, OtherPotassium IonophorePPAR, Non-SelectivePPARαPPARδPPARγPPARPregnane X ReceptorsPrion ProteinProgesterone ReceptorsProstacyclinProstaglandinProstanoid ReceptorsProtease-Activated ReceptorsProteasesProteasomeProteinasesProtein Kinase, Broad SpectrumProtein Kinase AProtein Kinase BProtein Kinase CProtein Kinase DProtein Kinase GProtein Ser/Thr PhosphatasesProtein SynthesisProtein Translocation, Exocytosis and EndocytosisProtein Tyrosine PhosphatasesPrP-ResPTH ReceptorsPTPPurine TransportersPyrimidine Transporters
S1P ReceptorssAHP ChannelsSAPKsTocriscreen Compound Library CollectionsSec7SecretaseSecretase, γ-Secretin ReceptorsSelectinsSensory Neuron-Specific ReceptorsSERCASerine ProteaseSerotonin (5-HT1) ReceptorsSerotonin (5-HT1A) ReceptorsSerotonin (5-HT1B) ReceptorsSerotonin (5-HT1D) ReceptorsSerotonin (5-ht1E) ReceptorsSerotonin (5-HT1F) ReceptorsSerotonin (5-HT2) ReceptorsSerotonin (5-HT2A) ReceptorsSerotonin (5-HT2B) ReceptorsSerotonin (5-HT2C) ReceptorsSerotonin (5-HT3) ReceptorsSerotonin (5-HT4) ReceptorsSerotonin (5-ht5) ReceptorsSerotonin (5-HT6) ReceptorsSerotonin (5-HT7) ReceptorsSerotonin N-acetyl transferaseSerotonin ReceptorsSerotonin RelatedSerotonin TransportersSerotonin UptakeSERTSF-1sGCShp1Shp2Sigma, General
Sigma1 ReceptorsSigma2 ReceptorsSigma ReceptorsSignal Transducers and Activators of TranscriptionSignal TransductionSir2-like Family DeacetylasesSirtuinSmoothened ReceptorsSmo ReceptorsSNSRSOC ChannelsSodium (Epithelial) ChannelsSodium (NaV) ChannelsSodium, Potassium, Chloride CotransporterSodium/Calcium ExchangerSodium ChannelsSomatostatin (sst) ReceptorsSpermidine acetyltransferaseSpermine acetyltransferaseSphingosine-1-Phosphate ReceptorsSphingosine KinaseSphingosine N-acyltransferasesPLA2Src Kinasesst ReceptorsSTATStem CellsSteroid Hormone ReceptorsSteroidogenic Factor-1STIM-Orai ChannelsStore Operated Calcium ChannelsStress-Activated Protein KinaseSyk KinaseSynthases, OtherSynthases/SynthetasesSynthetaseSynthetases, Other
T-Type Calcium ChannelsTachykinin, Non-SelectiveTachykinin NK1 ReceptorsTachykinin NK2 ReceptorsTachykinin NK3 ReceptorsTachykinin ReceptorsTankyraseTauTelomeraseTGF-β ReceptorsThrombinThromboxane A2 Synthetase Thromboxane ReceptorsThymidylate SynthetaseThyrotropin-Releasing Hormone ReceptorsTLRTNF-αToll-like Receptors
TopoisomeraseTP ReceptorsTranscription FactorsTransferasesTransforming Growth Factor Beta ReceptorsTransient Receptor Potential ChannelsTransportersTRH ReceptorsTriphosphoinositol ReceptorsTrk ReceptorsTRP ChannelsTRP Channels, OtherTRPVTrypsinTryptaseTryptophan HydroxylaseTubulinTumor Necrosis Factor-α
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