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Estrogen Receptors
More Information »Estrogen controls many cellular processes including growth, differentiation and function of the reproductive system. Estrogen is also responsible for the growth and maintenance of the skeleton and the normal function of the cardiovascular and nervous systems.
Estrogen Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 1417 | Daidzein |
| Estrogen receptor agonist. Also induces cell cycle arrest | |
| 1494 | DPN |
| Highly potent ERβ agonist | |
| 4494 |
(R)-DPN
|
| Enantiomer of DPN (Cat. No. 1494) | |
| 2266 | DY131 |
| Agonist selective for estrogen-related receptors ERRβ and ERRγ | |
| 4276 | ERB 041 |
| Potent ERβ agonist | |
| 2823 | α-Estradiol |
| Endogenous estrogen receptor agonist | |
| 2824 | β-Estradiol |
| Endogenous ER agonist | |
| 3588 | Estropipate |
| Estrogen receptor agonist and OATP1B1 inhibitor | |
| 3523 | FERb 033 |
| Potent and selective ERβ agonist | |
| 3075 | GSK 4716 |
| Selective ERRγ and ERRβ agonist | |
| 3819 | Liquiritigenin |
| Selective ERβ agonist | |
| 1426 | PPT |
| Subtype-selective ERα agonist | |
| 3366 | WAY 200070 |
| Selective ERβ agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 1047 | ICI 182,780 |
| Estrogen receptor antagonist | |
| 1991 | MPP dihydrochloride |
| Highly selective ERα antagonist | |
| 2662 | PHTPP |
| Selective ERβ antagonist | |
| 3928 | XCT 790 |
| Selective ERRα antagonist/inverse agonist | |
| 2183 | ZK 164015 |
| Potent estrogen receptor antagonist | |
Modulators |
|
Cat.No. |
Product Name / Activity |
| 3999 | Cyclofenil |
| Selective estrogen receptor modulator (SERM) | |
| 2280 | Raloxifene hydrochloride |
| Selective estrogen receptor modulator (SERM) | |
| 2676 | Y 134 |
| Selective estrogen receptor modulator (SERM), selective for ERα | |
Inhibitors |
|
Cat.No. |
Product Name / Activity |
| 4382 | Letrozole |
| Potent, reversible non-steroidal aromatase inhibitor | |
Other |
|
Cat.No. |
Product Name / Activity |
| 3388 | Anastrozole |
| Potent aromatase (CYP19) inhibitor | |
| 0743 | DPPE fumarate |
| Ligand for anti-estrogen binding site | |
| 3705 | Endoxifen |
| Potent antiestrogen; ERα ligand | |
| 1110 | Genistein |
| Estrogen receptor ligand. Also tyrosine kinase inhibitor | |
| 3224 | RU 58668 |
| Pure antiestrogen | |
| 0999 | Tamoxifen citrate |
| Estrogen receptor partial agonist/antagonist | |
| 1990 | (R,R)-THC |
| Potent subtype-selective ligand; ERα agonist/ERβ antagonist | |
| 3278 | YM 511 |
| Potent aromatase (CYP19) inhibitor | |
| 3975 | Zearalenone |
| Estrogen receptor ligand; mycotoxin | |
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Cancer Research Guide
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Nuclear Receptors Product Listing
Highlights over 150 products for nuclear receptors. Reserve your free copy today and be amongst the first to receive it.
Estrogen Pathway
Estrogen controls many cellular processes including growth, differentiation and function of the reproductive system. View pathway or download PDF today.
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