R&D Systems Inc. Tocris Bioscience Boston Biochem

Estrogen and Related Receptors

More Information »Estrogen controls many cellular processes including growth, differentiation and function of the reproductive system. Estrogen is also responsible for the growth and maintenance of the skeleton and the normal function of the cardiovascular and nervous systems.

Estrogen and Related Receptor Products

Agonists
Cat.No.
Product Name / Activity
1417 Daidzein
Estrogen receptor agonist. Also induces cell cycle arrest
1494 DPN
Highly potent ERβ agonist
4494 (R)-DPN
Enantiomer of DPN (Cat. No. 1494)
2266 DY131
Agonist selective for estrogen-related receptors ERRβ and ERRγ
4276 ERB 041
Potent ERβ agonist
2823 α-Estradiol
Endogenous estrogen receptor agonist
2824 β-Estradiol
Endogenous ER agonist
3588 Estropipate
Estrogen receptor agonist and OATP1B1 inhibitor
3523 FERb 033
Potent and selective ERβ agonist
3075 GSK 4716
Selective ERRγ and ERRβ agonist
3819 Liquiritigenin
Selective ERβ agonist
1426 PPT
Subtype-selective ERα agonist
3366 WAY 200070
Selective ERβ agonist
Antagonists
Cat.No.
Product Name / Activity
1047 ICI 182,780
Estrogen receptor antagonist
1991 MPP dihydrochloride
Highly selective ERα antagonist
2662 PHTPP
Selective ERβ antagonist
3928 XCT 790
Selective ERRα antagonist/inverse agonist
2183 ZK 164015
Potent estrogen receptor antagonist
Modulators
Cat.No.
Product Name / Activity
3999 Cyclofenil
Selective estrogen receptor modulator (SERM)
3412 (Z)-4-Hydroxytamoxifen
Metabolite of tamoxifen (Cat. No. 0999)
2280 Raloxifene hydrochloride
Selective estrogen receptor modulator (SERM)
0999 Tamoxifen citrate
Estrogen receptor partial agonist/antagonist
2676 Y 134
Selective estrogen receptor modulator (SERM), selective for ERα
Inhibitors
Cat.No.
Product Name / Activity
4382 Letrozole
Potent, reversible non-steroidal aromatase inhibitor
Other
Cat.No.
Product Name / Activity
3388 Anastrozole
Potent aromatase (CYP19) inhibitor
0743 DPPE fumarate
Ligand for anti-estrogen binding site
3705 Endoxifen
Potent antiestrogen; ERα ligand
1110 Genistein
Estrogen receptor ligand. Also tyrosine kinase inhibitor
3224 RU 58668
Pure antiestrogen
1990 (R,R)-THC
Potent subtype-selective ligand; ERα agonist/ERβ antagonist
3278 YM 511
Potent aromatase (CYP19) inhibitor
3975 Zearalenone
Estrogen receptor ligand; mycotoxin
Related Categories

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Bio-Techne Events

FEBS-EMBO 2014 Meeting

FEBS-EMBO 2014

August 30 - September 4, 2014

Paris, France

Booth Number: 22